Product apis-epigentics

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Catalog	name	Description	price
R-C-2701	GSK 525768A CAS：1260530-25-3	GSK 525768A is the enantiomer compound of GSK 525762A,which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2,Brd3,and Brd4);GSK 525768A has NO activity towards BET.	price>
R-C-2702	GSK1324726A (I-BET726) CAS：1300031-52-0	GSK1324726A is a novel,potent,and selective inhibitor of BET proteins with high affinity to BRD2(IC50=41nM),BRD3(IC50=31nM),and BRD4(IC50=22nM).	price>
R-C-2705	EPZ004777 CAS：1338466-77-5	EPZ004777 is a potent,selective DOT1L inhibitor with IC50 of 0.4nM in a cell-free assay and demonstrates>1,200-fold selectivity for DOT1L over all other tested PMTs.EPZ004777 induces apoptosis.	price>
R-C-2707	OG-L002 CAS:1357302-64-7	OG-L002 is a potent and highly selective LSD1 inhibitor with an IC50 of 0.02 μM.OG-L002 is a potent monoamine oxidases(MAO)inhibitor with IC50s of 1.38μM and 0.72μM for MAO-A and MAO-B,respectively.OG-L002 potently inhibits the expression of HSV IE genes.	price>
R-C-2708	CBB1003 CAS:1379573-88-2	CBB1003 is a novel histone demethylase LSD1 inhibitor with IC50 of 10.54uM.	price>
R-C-2709	CBB1007 CAS:1379573-92-8	CBB1007 is a cell-permeable amidino-guanidinium compound that acts as a potent,reversible and substrate competitive LSD1 selective inhibitor (IC50=5.27μM for hLSD1).	price>
R-C-2710	YM 750 CAS:138046-43-2	YM-750 is a potent acyl-CoA:cholesterol acyltransferase(ACAT)inhibitor(IC50=0.18 μM).ACAT catalyzes the formation of cholesteryl esters from cholesterol and long-chain fatty-acyl-coenzyme A.	price>
R-C-2711	GSK J5 CAS:1394854-51-3	Inactive isomer of GSK J4;also cell permeable ester derivative of the inactive control,GSK J2.	price>

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