Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3541	DPTN dihydrochloride CAS No.325767-87-1	DPTN/CAS No.325767-87-1 is a potent and selective human, mouse, and rat A3AR antagonist with Ki values of 1.65, 9.61, and 8.53 nM, respectively.	price>
R-R-3542	M1069	M1069 is a selective and orall active, dual A2A/A2B adenosine receptor antagonist with a selectivity of >100 fold against the A1 and A3 receptors. M1069 counteracts immune-suppressive mechanisms of adenosine, and exhibits anti-tumor activity.	price>
R-R-3543	MIPS521 CAS No.1146188-19-3	MIPS521/CAS No.1146188-19-3 is a positive allosteric modulator of adenosine A1 receptor (A1AR). MIPS521 also has a lower A1R allosteric affinity (pKB=4.95; KB=11 μM). MIPS521 exhibits pain-relieving effects in vivo through modulation of the increased levels of endogenous adenosine.	price>
R-R-3544	N-[(4-Aminophenyl)methyl]adenosine CAS No.95523-13-0	N-[(4-Aminophenyl)methyl]adenosine/CAS No.95523-13-0 is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5-Nucleotidase.	price>
R-R-3545	Trabodenoson CAS No.871108-05-3	Trabodenoson (INO-8875)/CAS No.871108-05-3, an adenosine mimetic, is a highly selective Adenosine A1 receptor agonist. Trabodenoson (INO-8875) is used in the study for Primary Open-Angle Glaucoma.	price>
R-R-3546	Adenosine amine congener CAS No.96760-69-9	Adenosine amine congener (ADAC)/CAS No.96760-69-9 is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. Adenosine amine congener also has neuroprotective effects.	price>
R-R-3547	MRS1220 CAS No.183721-15-5	MRS1220/CAS No.183721-15-5, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of diseases of the central nervous system. MRS1220 reduces glioblastoma tumor size and blood vessel formation in vivo.	price>
R-R-3548	PSB36 CAS No.524944-72-7	PSB36/CAS No.524944-72-7 is a potent and selective antagonist of adenosine A1 receptor, with Kis 0.12 nM, 187 nM, 552 nM, 2300 nM, and 6500 nM for rA1, hA2B, rA2A, hA3 and rA3 receptors respectively. PSB36 can be used for the research of hyperalgesia.	price>
R-R-3549	Theophylline-d6 CAS No.117490-39-8	Theophylline-d6/CAS No.117490-39-8 is the deuterium labeled Theophylline. Theophylline is a nonselective phosphodiesterase (PDE) inhibitor, adenosine receptor blocker, and histone deacetylase (HDAC) activator.	price>
R-R-3550	LUF6000 CAS No.890087-21-5	LUF6000/CAS No.890087-21-5 is an orally active allosteric modulator of the A3 adenosine receptor. LUF6000 has potent anti-inflammatory effect.	price>

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