Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3543	MIPS521 CAS No.1146188-19-3	MIPS521/CAS No.1146188-19-3 is a positive allosteric modulator of adenosine A1 receptor (A1AR). MIPS521 also has a lower A1R allosteric affinity (pKB=4.95; KB=11 μM). MIPS521 exhibits pain-relieving effects in vivo through modulation of the increased levels of endogenous adenosine.	price>
R-R-3544	N-[(4-Aminophenyl)methyl]adenosine CAS No.95523-13-0	N-[(4-Aminophenyl)methyl]adenosine/CAS No.95523-13-0 is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5-Nucleotidase.	price>
R-R-3545	Trabodenoson CAS No.871108-05-3	Trabodenoson (INO-8875)/CAS No.871108-05-3, an adenosine mimetic, is a highly selective Adenosine A1 receptor agonist. Trabodenoson (INO-8875) is used in the study for Primary Open-Angle Glaucoma.	price>
R-R-3546	Adenosine amine congener CAS No.96760-69-9	Adenosine amine congener (ADAC)/CAS No.96760-69-9 is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. Adenosine amine congener also has neuroprotective effects.	price>
R-R-3547	MRS1220 CAS No.183721-15-5	MRS1220/CAS No.183721-15-5, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of diseases of the central nervous system. MRS1220 reduces glioblastoma tumor size and blood vessel formation in vivo.	price>
R-R-3548	PSB36 CAS No.524944-72-7	PSB36/CAS No.524944-72-7 is a potent and selective antagonist of adenosine A1 receptor, with Kis 0.12 nM, 187 nM, 552 nM, 2300 nM, and 6500 nM for rA1, hA2B, rA2A, hA3 and rA3 receptors respectively. PSB36 can be used for the research of hyperalgesia.	price>
R-R-3549	Theophylline-d6 CAS No.117490-39-8	Theophylline-d6/CAS No.117490-39-8 is the deuterium labeled Theophylline. Theophylline is a nonselective phosphodiesterase (PDE) inhibitor, adenosine receptor blocker, and histone deacetylase (HDAC) activator.	price>
R-R-3550	LUF6000 CAS No.890087-21-5	LUF6000/CAS No.890087-21-5 is an orally active allosteric modulator of the A3 adenosine receptor. LUF6000 has potent anti-inflammatory effect.	price>
R-R-3551	A2B receptor antagonist 2 CAS No.784-90-7	A2B receptor antagonist 2 (compound 18)/CAS No.784-90-7 is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively.	price>
R-R-3552	PSB 0777 ammonium hydrate	PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist with Ki values of 44.4 nM, 360 nM for rat and human A2A receptors, respectively. PSB 0777 ammonium hydrate has Ki values of ≥10000 nM, 541 nM for rat and human A1 receptors, respectively. PSB 0777 ammonium hydrate shows poor brain penetrant and perorally non-absorbable effect. PSB 0777 ammonium hydrate has the potential for inflammatory bowel disease (IBS) research research.	price>

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