Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3551	A2B receptor antagonist 2 CAS No.784-90-7	A2B receptor antagonist 2 (compound 18)/CAS No.784-90-7 is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively.	price>
R-R-3552	PSB 0777 ammonium hydrate	PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist with Ki values of 44.4 nM, 360 nM for rat and human A2A receptors, respectively. PSB 0777 ammonium hydrate has Ki values of ≥10000 nM, 541 nM for rat and human A1 receptors, respectively. PSB 0777 ammonium hydrate shows poor brain penetrant and perorally non-absorbable effect. PSB 0777 ammonium hydrate has the potential for inflammatory bowel disease (IBS) research research.	price>
R-R-3553	ANR94 CAS No.634924-89-3	ANR94/CAS No.634924-89-3 is a potent and selective adenosine A2A receptor (AA2AR) antagonist with an Ki of 46 nM for hAA2AR. ANR94 has the potential for the research of Parkinson disease.	price>
R-R-3554	Xanthine amine congener hydrochloride CAS No.1783977-95-6	Xanthine amine congener (XAC) hydrochloride/CAS No.1783977-95-6 is a non-selective adenosine receptor antagonist. Xanthine amine congener hydrochloride induces convulsions in mice.	price>
R-R-3555	MRS1334 CAS No.192053-05-7	MRS1334/CAS No.192053-05-7 is a potent and selective human adenosine A3 receptor antagonist with Kis of 2.69 nM, >100 nM, >100 nM for hA3, rA1, rA2A, respectively. MRS1334 blocks the protective effect of Cl-IB-MECA leading to significant bradycardia and elevated ST segment. MRS1334 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-R-3556	8-Cyclopentyl-1,3-dimethylxanthine CAS No.35873-49-5	8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a)/CAS No.35873-49-5 is a selective adenosine A1 receptor antagonist with Kis of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively.	price>
R-R-3557	Norisoboldine CAS No.23599-69-1	Norisoboldine/CAS No.23599-69-1 is an orally active natural aryl hydrocarbon receptor (AhR) agonist. Norisoboldine, as a major isoquinoline alkaloid present in Radix Linderae, can be used for the research of Rheumatoid arthritis and Ulcerative colitis.	price>
R-R-3558	Cirazoline hydrochloride CAS No.40600-13-3	Cirazoline hydrochloride (LD 3098 hydrochloride)/CAS No.40600-13-3 is a potent competitive full α1A-adrenergic receptor (α1A-AR) agonist (Ki=120 nM) and only a partial agonist at α1B-AR (Ki= 960 nM) and α1D-AR (Ki=660 nM).	price>
R-R-3559	MRS-3777 hemioxalate CAS No.1186195-57-2	MRS-3777 hemioxalate/CAS No.1186195-57-2 is a selective adenosine A3 receptor antagonist.	price>
R-R-3560	Adenosine receptor antagonist 2 CAS No.2703054-47-9	Adenosine receptor antagonist 2/CAS No.2703054-47-9 is an orally active A2a/A2b adenosine receptor antagonist with IC50s of 1 nM and 3 nM, respectively. Adenosine receptor antagonist 2 has anti-tumor activity.	price>

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