Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3553	ANR94 CAS No.634924-89-3	ANR94/CAS No.634924-89-3 is a potent and selective adenosine A2A receptor (AA2AR) antagonist with an Ki of 46 nM for hAA2AR. ANR94 has the potential for the research of Parkinson disease.	price>
R-R-3554	Xanthine amine congener hydrochloride CAS No.1783977-95-6	Xanthine amine congener (XAC) hydrochloride/CAS No.1783977-95-6 is a non-selective adenosine receptor antagonist. Xanthine amine congener hydrochloride induces convulsions in mice.	price>
R-R-3555	MRS1334 CAS No.192053-05-7	MRS1334/CAS No.192053-05-7 is a potent and selective human adenosine A3 receptor antagonist with Kis of 2.69 nM, >100 nM, >100 nM for hA3, rA1, rA2A, respectively. MRS1334 blocks the protective effect of Cl-IB-MECA leading to significant bradycardia and elevated ST segment. MRS1334 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-R-3556	8-Cyclopentyl-1,3-dimethylxanthine CAS No.35873-49-5	8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a)/CAS No.35873-49-5 is a selective adenosine A1 receptor antagonist with Kis of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively.	price>
R-R-3557	Norisoboldine CAS No.23599-69-1	Norisoboldine/CAS No.23599-69-1 is an orally active natural aryl hydrocarbon receptor (AhR) agonist. Norisoboldine, as a major isoquinoline alkaloid present in Radix Linderae, can be used for the research of Rheumatoid arthritis and Ulcerative colitis.	price>
R-R-3558	Cirazoline hydrochloride CAS No.40600-13-3	Cirazoline hydrochloride (LD 3098 hydrochloride)/CAS No.40600-13-3 is a potent competitive full α1A-adrenergic receptor (α1A-AR) agonist (Ki=120 nM) and only a partial agonist at α1B-AR (Ki= 960 nM) and α1D-AR (Ki=660 nM).	price>
R-R-3559	MRS-3777 hemioxalate CAS No.1186195-57-2	MRS-3777 hemioxalate/CAS No.1186195-57-2 is a selective adenosine A3 receptor antagonist.	price>
R-R-3560	Adenosine receptor antagonist 2 CAS No.2703054-47-9	Adenosine receptor antagonist 2/CAS No.2703054-47-9 is an orally active A2a/A2b adenosine receptor antagonist with IC50s of 1 nM and 3 nM, respectively. Adenosine receptor antagonist 2 has anti-tumor activity.	price>
R-R-3561	Adenosine A1 receptor activator T62 CAS No.40312-34-3	Adenosine A1 receptor activator T62/CAS No.40312-34-3 is an allosteric enhancer of adenosine A1 receptor. Adenosine A1 receptor activator T62 produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve-injury pain.	price>
R-R-3562	Tecadenoson CAS No.204512-90-3	Tecadenoson (CVT-510)/CAS No.204512-90-3 is a selective A1 adenosine receptor agonist.	price>

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