Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3563	CV1808 CAS No.53296-10-9	CV1808 (2-Phenylaminoadenosine)/CAS No.53296-10-9 is a non-selective A2 adenosine receptor (A2 AR) agonist with Kis of 76 and 1450 nM for A2A and A3 adenosine receptor subtypes, respectively.	price>
R-R-3564	FR194921 CAS No.202646-80-8	FR194921/CAS No.202646-80-8 is a potent, selective and orally active and cross the blood-brain barrier Adenosine A1 antagonist with Ki value of 6.6, 5400 nM for A1, A2A, respectively. FR194921 shows cognitive-enhancing and anxiolytic activity.	price>
R-R-3565	HEMADO CAS No.403842-38-6	HEMADO/CAS No.403842-38-6 is a potent and selective adenosine A3 receptor agonist with a Ki of 1.1 nM at the human A3 subtype. HEMADO is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-R-3566	MRE3008F20 CAS No.252979-43-4	MRE3008F20/CAS No.252979-43-4 is a highly potent and selective adenosine A3 receptor (AA3R) antagonist that inhibits agonist-induced cAMP elevation in resting T cells with an IC50 of 5 nM.	price>
R-C-1867	JNJ-46778212(VU 0409551) CAS:1363281-27-9	JNJ-46778212(VU 0409551)is an mGlu5 positive allosteric modulator with an EC50 of 260nM.	price>
R-R-3567	VUF-5574 CAS No.280570-45-8	VUF-5574/CAS No.280570-45-8 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.	price>
R-R-3568	Enprofylline CAS No.41078-02-8	Enprofylline/CAS No.41078-02-8 acts as a selective and competitive A2B receptor antagonist with the Ki of 7 μM. Enprofylline also acts as a phosphodiesterase inhibitor. Enprofylline can be used for the research of asthma, chronic obstructive pulmonary disease.	price>
R-R-3569	KI-7 CAS No.1489263-00-4	KI-7/CAS No.1489263-00-4 is an A2B adenosine receptor positive allosteric modulator. KI-7 potentiates the cAMP accumulation induced by the non-selective A2B adenosine receptor agonist NECA (EC50=445.8 nM). KI-7 also potentiates the cAMP accumulation induced by the selective A2B adenosine receptor agonist BAY 60-6583 as well as by adenosine with EC50s of 2390 nM and 2550 nM, respectively.	price>
R-R-3570	Doxofylline-d6 CAS No.1219805-99-8	Doxofylline-d6/CAS No.1219805-99-8 is the deuterium labeled Doxofylline. Doxofylline is an antagonist of adenosine A1 receptor which also inhibits phosphodiesterase IV.	price>
R-R-3571	LUF6096 CAS No.1116652-18-6	LUF6096/CAS No.1116652-18-6, a potent allosteric enhancer of the adenosine A3 receptor, is able to allosterically enhance agonist binding. LUF6096 shows low orthosteric affinity for any of the adenosine receptors. LUF6096 shows protective effects in myocardial ischemia/reperfusion injury.	price>

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