Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3561	Adenosine A1 receptor activator T62 CAS No.40312-34-3	Adenosine A1 receptor activator T62/CAS No.40312-34-3 is an allosteric enhancer of adenosine A1 receptor. Adenosine A1 receptor activator T62 produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve-injury pain.	price>
R-R-3562	Tecadenoson CAS No.204512-90-3	Tecadenoson (CVT-510)/CAS No.204512-90-3 is a selective A1 adenosine receptor agonist.	price>
R-R-3563	CV1808 CAS No.53296-10-9	CV1808 (2-Phenylaminoadenosine)/CAS No.53296-10-9 is a non-selective A2 adenosine receptor (A2 AR) agonist with Kis of 76 and 1450 nM for A2A and A3 adenosine receptor subtypes, respectively.	price>
R-R-3564	FR194921 CAS No.202646-80-8	FR194921/CAS No.202646-80-8 is a potent, selective and orally active and cross the blood-brain barrier Adenosine A1 antagonist with Ki value of 6.6, 5400 nM for A1, A2A, respectively. FR194921 shows cognitive-enhancing and anxiolytic activity.	price>
R-R-3565	HEMADO CAS No.403842-38-6	HEMADO/CAS No.403842-38-6 is a potent and selective adenosine A3 receptor agonist with a Ki of 1.1 nM at the human A3 subtype. HEMADO is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-R-3566	MRE3008F20 CAS No.252979-43-4	MRE3008F20/CAS No.252979-43-4 is a highly potent and selective adenosine A3 receptor (AA3R) antagonist that inhibits agonist-induced cAMP elevation in resting T cells with an IC50 of 5 nM.	price>
R-C-1867	JNJ-46778212(VU 0409551) CAS:1363281-27-9	JNJ-46778212(VU 0409551)is an mGlu5 positive allosteric modulator with an EC50 of 260nM.	price>
R-R-3567	VUF-5574 CAS No.280570-45-8	VUF-5574/CAS No.280570-45-8 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.	price>
R-R-3568	Enprofylline CAS No.41078-02-8	Enprofylline/CAS No.41078-02-8 acts as a selective and competitive A2B receptor antagonist with the Ki of 7 μM. Enprofylline also acts as a phosphodiesterase inhibitor. Enprofylline can be used for the research of asthma, chronic obstructive pulmonary disease.	price>
R-R-3569	KI-7 CAS No.1489263-00-4	KI-7/CAS No.1489263-00-4 is an A2B adenosine receptor positive allosteric modulator. KI-7 potentiates the cAMP accumulation induced by the non-selective A2B adenosine receptor agonist NECA (EC50=445.8 nM). KI-7 also potentiates the cAMP accumulation induced by the selective A2B adenosine receptor agonist BAY 60-6583 as well as by adenosine with EC50s of 2390 nM and 2550 nM, respectively.	price>

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