Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3513	ML 10302 hydrochloride CAS No.186826-17-5	ML 10302 hydrochloride/CAS No.186826-17-5 is a potent and selective 5-HT4 receptor agonist, with an EC50 of 4 nM. ML 10302 hydrochloride displays more than 680-fold selectivity over 5-HT3 receptor in binding assay.	price>
R-R-3514	5-HT4 antagonist 1 CAS No.261766-73-8	5-HT4 antagonist 1/CAS No.261766-73-8 is a 5-HT4 receptor antagonist with a pKi of 9.6.	price>
R-R-3515	AL-34662 CAS No.210580-75-9	AL-34662/CAS No.210580-75-9 is a selective 5-HT2A receptoragonist (IC50: 0.77 nM and 1.5 nM for rat and human 5-HT2 receptor). AL-34662 is also a weak α-1D adrenergic agonist activity (EC50:0.4 μM). AL-34662 is an ocular hypotensive agent.	price>
R-R-3516	RS 23597-190 CAS No.149719-06-2	RS 23597-190 (EP-A-501322)/CAS No.149719-06-2 is a high affinity and selective 5-HT4 receptor antagonist. RS 23597-190 inhibits 5-HT-induced tachycardia. RS 23597-190 significantly inhibits superoxide production in high glucose.	price>
R-R-3517	CGS 21680 Hydrochloride CAS No.124431-80-7	CGS 21680 Hydrochloride/CAS No.124431-80-7 is a selective adenosine A2A receptor agonist with a Ki of 27 nM.	price>
R-R-3518	Istradefylline CAS No.155270-99-8	Istradefylline/CAS No.155270-99-8 is a very potent, selective and orally active adenosine A2A receptor antagonist with Ki of 2.2 nM in experimental models of Parkinson disease.	price>
R-R-3519	SCH-202676 hydrobromide CAS No.265980-25-4	SCH-202676 hydrobromide/CAS No.265980-25-4 is an allosteric modulator of G protein-coupled receptors (GPCRs) and adenosine receptor (AR). SCH-202676 hydrobromide has antiviral activity and inhibits 3CLpro in a time-dependent manner with an IC50 value of 0.655 μM.	price>
R-R-3520	BAY 60-6583 CAS No.910487-58-0	BAY 60-6583/CAS No.910487-58-0 is a potent and high-affinity agonist of adenosine A2B receptor (EC50 = 3 nM) over A1, A2A, and A3 receptors. BAY 60-6583 binds to mouse, rabbit, and dog A2BAR with Ki values of 750 nM, 340 nM and 330 nM, respectively. BAY 60-6583 has a cardioprotective effect in a myocardial ischemia model.	price>
R-R-3521	DPCPX CAS No.102146-07-6	DPCPX (PD 116948)/CAS No.102146-07-6, a xanthine derivative, is a highly potent and selective Adenosine A1 receptor antagonist, with a Ki of 0.46 nM in 3H-CHA binding to A1 receptors in rat whole brain membranes.	price>
R-R-3522	MRS 1754 CAS No.264622-58-4	MRS 1754/CAS No.264622-58-4 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats.	price>

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