Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-C-1765	Treprostinil (LRX-15) CAS：81846-19-7	Treprostinil(LRX-15)is a potent DP1 and EP2 agonist with EC50 values of 0.6±0.1 and 6.2±1.2nM,respectively.	price>
R-C-1766	Pitolisant CAS:362665-56-3	Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor(Ki=0.16nM).	price>
R-C-1770	Amiselimod hydrochloride CAS:942398-84-7	Amiselimod hydrochloride is a novel sphingosine 1-phosphate receptor-1(S1P1) modulator,designed to reduce the bradycardia effects associated with fingolimod and other S1P receptor modulators.	price>
R-C-1771	SB408124 CAS:288150-92-5	SB-408124 is a selective non-peptide orexin OX1 receptor antagonist(Kb values are 21.7 and 1405 nM for human OX1 and OX2 receptors respectively).Blocks orexin-A induced grooming following oral administration in vivo.	price>
R-R-3477	Ondansetron-d5 CAS No.1219798-86-3	Ondansetron-d5/CAS No.1219798-86-3 is the deuterium labeled Ondansetron. Ondansetron (GR 38032; SN 307) is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy.	price>
R-R-3478	Ziprasidone-d8 CAS No.1126745-58-1	Ziprasidone-d8/CAS No.1126745-58-1 is deuterium labeled Ziprasidone, which is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity.	price>
R-R-3479	AP521 CAS No.151227-08-6	AP521/CAS No.151227-08-6 is an agonist of human 5-HT1A receptor with an IC50 of 94 nM.	price>
R-R-3480	Vilazodone-d8 CAS No.1794789-93-7	Vilazodone-d8/CAS No.1794789-93-7 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist.	price>
R-R-3481	H-9 Dihydrochloride CAS No.116700-36-8	H-9 Dihydrochloride/CAS No.116700-36-8 is a PKA (protein kinase) inhibitor. H-9 Dihydrochloride (10 μM) significantly reduces the excitatory response to 5-HT. H-9 Dihydrochloride also has a direct effect on pharyngeal activity. H-9 Dihydrochloride inhibits signal-transduction and cell growth in EGF (epidermal growth factor)-dependent epithelial cell lines.	price>
R-R-3482	(S)-Mirtazapine-d3	(S)-Mirtazapine-d3 is a deuterium labeled (S)-Mirtazapine. (S)-Mirtazapine is a S(+)-enantiomer of Mirtazapine with pronociceptive properties in an animal model of acute thermal nociception.(S)-Mirtazapine is a stereoselective 5-HT2 receptor antagonist. (S)-Mirtazapine is metabolized by CYP2D6 and CYP1A2.	price>

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