Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3419	Cyclobenzaprine-d3 hydrochloride CAS No.1184983-42-3	Cyclobenzaprine-d3 (hydrochloride)/CAS No.1184983-42-3 is the deuterium labeled Cyclobenzaprine hydrochloride. Cyclobenzaprine hydrochloride (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant.	price>
R-R-3420	LY 344864 S-enantiomer CAS No.186544-27-4	LY 344864 S-enantiomer/CAS No.186544-27-4 is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist.	price>
R-R-3421	Perphenazine-d4 CAS No.155593-75-2	Perphenazine-d4/CAS No.155593-75-2 is the deuterium labeled Perphenazine. Perphenazine is a typical antipsychotic agent, inhibits 5-HT2Areceptor, Alpha-1A adrenergic receptor, Dopamine receptor D2/D3, D2L receptor, and Histamine H1 receptor, with Ki values of 5.6, 10, 0.765/0.13, 3.4, and 8 nM, respectively.	price>
R-R-3422	3-Hydroxy agomelatine-d3 CAS No.1079774-23-4	3-Hydroxy agomelatine-d3/CAS No.1079774-23-4 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is a 5-HT2C receptor antagonist with an IC50 of 3.2 μM and a Ki of 1.8 μM.	price>
R-R-3423	Eplivanserin (mixture) CAS No.130581-13-4	Eplivanserin mixture (SR-46349 mixture)/CAS No.130581-13-4 is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1.	price>
R-R-3424	3-AQC CAS No.201216-42-4	3-AQC/CAS No.201216-42-4, a piperazinylquinoxaline derivative, is a potent and competitive 5-HT3 receptor antagonist.	price>
R-R-3425	Ondansetron-13C,d3 CAS No.2699607-85-5	Ondansetron-13C,d3/CAS No.2699607-85-5 is the 13C- and deuterium labeled Ondansetron.	price>
R-R-3426	Brexpiprazole-d8 CAS No.1427049-21-5	Brexpiprazole-d8/CAS No.1427049-21-5 is a deuterium labeled Brexpiprazole (OPC-34712). Brexpiprazole, an atypical antipsychotic agent, is a partial agonist of human 5-HT1A and dopamine receptor (Ki=0.12 nM and 0.3 nM, respectively). Brexpiprazole is also a 5-HT2A receptor antagonist (Ki=0.47 nM).	price>
R-R-3427	Agomelatin-d3 CAS No.1079389-38-0	Agomelatin-d3/CAS No.1079389-38-0 is the deuterium labeled Agomelatine. Agomelatine (S-20098) is a specific agonist of MT1 and MT2 receptors with Kis of 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and HEK-hMT2, respectively. Agomelatine is a selective 5-HT2C receptor antagonist with pKis of 6.4 and 6.2 at native (porcine) and cloned, human 5-HT2C receptors, respectively.	price>
R-R-3428	Cinitapride CAS No.66564-14-5	Cinitapride/CAS No.66564-14-5 is a nonselective 5-HT1 and 5-HT4 receptors agonist and a 5-HT2 and D2 antagonist. Cinitapride can be used in functional dyspepsia (FD) and gastroesophageal reflux disease (GERD) research.	price>

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