Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3397	Aripiprazole (1,1,2,2,3,3,4,4-d8) CAS No.1089115-04-7	Aripiprazole (1,1,2,2,3,3,4,4-d8)/CAS No.1089115-04-7 is the deuterium labeled Aripiprazole. Aripiprazole (OPC-14597) is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.	price>
R-R-3398	Paliperidone-d4 CAS No.1020719-55-4	Paliperidone-d4/CAS No.1020719-55-4 is the deuterium labeled Paliperidone. Paliperidone (9-Hydroxyrisperidone), the major active metabolite of Risperidone, is a dopamine D2 antagonist and 5-HT2A antagonist. Paliperidone is also active as an antagonist at α1 and α2 adrenergic receptors and H1-histaminergic receptors. Paliperidone, a antipsychotic agent, shows efficacy against schizophrenia.	price>
R-R-3399	Alverine-d5 citrate CAS No.1215327-00-6	Alverine-d5 (citrate)/CAS No.1215327-00-6 is the deuterium labeled Alverine citrate.	price>
R-R-3400	Trazodone-d6 hydrochloride CAS No.1181578-71-1	Trazodone-d6 (hydrochloride)/CAS No.1181578-71-1 is the deuterium labeled Trazodone hydrochloride.	price>
R-R-3401	MS 245 oxalate CAS No.275363-58-1	MS 245 oxalate/CAS No.275363-58-1 is a potent antagonist of 5-HT6 receptor with a Ki of 2 nM.	price>
R-R-3402	Blonanserin-d5 CAS No.1346599-86-7	Blonanserin-d5/CAS No.1346599-86-7 is a deuterium labeled Blonanserin. Blonanserin is a dopamine D2/5-HT2 receptor antagonist and an atypical antipsychotic.	price>
R-R-3403	SB-216641A CAS No.193611-67-5	SB-216641A (SB-216641 hydrochloride)/CAS No.193611-67-5 is a selective antagonist of 5-HT1B/D receptor. SB-216641A shows high affinity and selectivity for h5-HT1B receptors over h5-HT1D receptors. SB-216641A inhibits the function of SKF-99101H.	price>
R-R-3404	Cyproheptadine-d3 CAS No.2712455-05-3	Cyproheptadine-d3/CAS No.2712455-05-3 is deuterium labeled Cyproheptadine.	price>
R-R-3405	Robalzotan hydrochloride CAS No.184674-99-5	Robalzotan hydrochloride (NAD-299 hydrochloride)/CAS No.184674-99-5 is a potent and selective 5-Hydroxytryptamine 1A (5-HT1A) inhibitor. Robalzotan hydrochloride increases the firing rate of 5-HT cells. Robalzotan hydrochloride induces 5-HT1A receptor occupancy. Robalzotan hydrochloride has the potential for the research of a cholinergic deficit in the central -nervous system.	price>
R-R-3406	(Rac)-Rotigotine CAS No.92206-54-7	(Rac)-Rotigotine (N-0437)/CAS No.92206-54-7 is a racemate of Rotigotine. Rotigotine is a full agonist of?dopamine receptor, a partial agonist of the?5-HT1A receptor, and an antagonist of the?α2B-adrenergic receptor, with?Kis of 0.71?nM, 4-15?nM, and 83?nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor.	price>

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