Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3390	(Rac)-Rotigotine hydrochloride CAS No.102120-99-0	(Rac)-Rotigotine hydrochloride/CAS No.102120-99-0 is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor, with Kis of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor.	price>
R-R-3391	Pardoprunox hydrochloride CAS No.269718-83-4	Pardoprunox (SLV-308) hydrochloride/CAS No.269718-83-4 is a partial dopamine D2 and D3 receptor partial agonist and a serotonin 5-HT1A receptor agonist, with pEC50s of 8, 9.2, and 6.3, respectively.	price>
R-R-3392	Isocorynoxeine CAS No.51014-29-0	Isocorynoxeine/CAS No.51014-29-0, an isorhynchophylline-related alkaloid, exhibits a dose-dependent inhibition of 5-HT2A receptor-mediated current response with an IC50 of 72.4 μM.	price>
R-R-3393	Lintopride CAS No.107429-63-0	Lintopride/CAS No.107429-63-0 is a 5HT4 antagonist with moderate 5HT3 antagonist properties.	price>
R-C-1694	GSK-189254 CAS：720690-73-3	GSK189254A(GSK189254)is a novel,potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively.	price>
R-R-3394	Lesopitron dihydrochloride CAS No.132449-89-9	Lesopitron dihydrochloride/CAS No.132449-89-9 is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes.	price>
R-R-3395	Lidanserin CAS No.73725-85-6	Lidanserin (ZK-33839)/CAS No.73725-85-6 acts as a 5-HT2A and α1-adrenergic receptor antagonist.	price>
R-R-3396	Sertindole-d4 CAS No.1794737-42-0	Sertindole-d4/CAS No.1794737-42-0 is the deuterium labeled Sertindole. Sertindole, a neuroleptic, is one of the newer antipsychotic medications available.	price>
R-R-3397	Aripiprazole (1,1,2,2,3,3,4,4-d8) CAS No.1089115-04-7	Aripiprazole (1,1,2,2,3,3,4,4-d8)/CAS No.1089115-04-7 is the deuterium labeled Aripiprazole. Aripiprazole (OPC-14597) is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.	price>
R-R-3398	Paliperidone-d4 CAS No.1020719-55-4	Paliperidone-d4/CAS No.1020719-55-4 is the deuterium labeled Paliperidone. Paliperidone (9-Hydroxyrisperidone), the major active metabolite of Risperidone, is a dopamine D2 antagonist and 5-HT2A antagonist. Paliperidone is also active as an antagonist at α1 and α2 adrenergic receptors and H1-histaminergic receptors. Paliperidone, a antipsychotic agent, shows efficacy against schizophrenia.	price>

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