Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3353	Velusetrag hydrochloride CAS No.866933-51-9	Velusetrag (TD-5108) hydrochloride/CAS No.866933-51-9 is an orally active, potent and selective agonist of serotonin 5-HT4 receptor (5-HT4R), with a pKi of 7.7. Velusetrag hydrochloride exhibits no affinity (Ki>10 μM) for 5-HT2A and 5-HT2B receptors.	price>
R-C-1654	Orexin 2 Receptor Agonist CAS：1796565-52-0	Orexin 2 Receptor Agonist is a potent(EC50 on OX2R is 23nM)and OX2R-selective (OX1R/OX2R EC50 ratio is 70) agonist.	price>
R-R-3354	Aripiprazole-d8 CAS No.1089115-06-9	Aripiprazole-d8/CAS No.1089115-06-9 is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.	price>
R-C-1655	piperoxan.HCl CAS: 135-87-5	Piperoxan hydrochloride(Benodaine,Fourneau 933,F933,DL-Piperoxan)is an antagonist of α2(alpha 2)adrenoceptor.	price>
R-C-1659	MK-1064 CAS：1207253-08-4	MK-1064 is a selective orexin 2 receptor antagonist(2-SORA)for the research of insomnia.	price>
R-C-1677	PF-04418948 CAS：1078166-57-0	PF-04418948 is a novel,potent and selective prostaglandin EP2 receptor antagonist.PF-04418948 inhibited prostaglandin E(2)(PGE(2))-induced increase in cAMP in cells expressing EP(2)receptors with a functional K(B)value of 1.8nM.	price>
R-R-3377	Facinicline hydrochloride CAS No.677305-02-1	Facinicline hydrochloride (RG3487 hydrochloride)/CAS No.677305-02-1 is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR. Facinicline hydrochloride (RG3487 hydrochloride) improves cognition and sensorimotor gating in rodents. Facinicline hydrochloride (RG3487 hydrochloride) shows high affinity (antagonist) to 5-HT3Rs with a Ki value of 1.2 nM.	price>
R-R-3378	Revexepride CAS No.219984-49-3	Revexepride/CAS No.219984-49-3 is a highly selective 5-HT4 receptor agonist, and a potential inducer of CYP3A4 enzyme, used for the treatment of gastroesophageal reflux disease.	price>
R-R-3379	Relenopride hydrochloride CAS No.1221416-42-7	Relenopride (YKP10811) hydrochloride/CAS No.1221416-42-7 is a specific and selective 5-HT4 receptor agonist (Ki=4.96 nM). Relenopride hydrochloride has 120-fold and 6-fold lower affinity, respectively, for 5-HT2A (Ki=600 nM) and 5-HT2B receptors (Ki=31 nM) than for 5-HT4. Relenopride hydrochloride increases gastrointestinal (GI) motility.	price>
R-C-1680	Carteolol hydrochloride CAS：51781-21-6	Carteolol hydrochloride(OPC-1085 hydrochloride)is a non-selective beta blocker used to treat glaucoma.	price>

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