Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3380	TC-2153 CAS No.1381769-23-8	TC-2153/CAS No.1381769-23-8 is a selective inhibitor of striatal-enriched protein tyrosine phosphatase (STEP), with psychotropic activity and low acute toxicity. TC-2153 increases the expression of brain-derived neurotropic factor (BDNF) in the brain. And it decreases MAOA and 5-HT1A receptors mRNA level in midbrain. TC-2153 also inhibits 5-HT2A receptor-mediated signaling.	price>
R-R-3381	(R)-Praziquantel-d11 CAS No.1399880-38-6	(R)-Praziquantel-d11/CAS No.1399880-38-6 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel, the active enantiomer of Praziquantel, is a partial agonist of the human 5-HT2B receptor. (R)-Praziquantel acts as an antischistosomal eutomer.	price>
R-C-1682	SQ22536 CAS：17318-31-9	SQ22536(9-(tetrahydrofuran-2-yl)-9h-purin-6-amine)is an inhibitor of adenylyl cyclase with an IC50 of 1.4μM.It can inhibit PGE1-stimulated increases in cAMP levels in intact human platelets.	price>
R-R-3382	Clozapine-d8 CAS No.1185053-50-2	Clozapine-d8/CAS No.1185053-50-2 is the deuterium labeled Clozapine. Clozapine is an antipsychotic used for the research of schizophrenia. Clozapine has high affinity for a number of neuroreceptors.	price>
R-R-3383	Ipsapirone CAS No.95847-70-4	Ipsapirone (TVX Q 7821)/CAS No.95847-70-4 is an anxiolytic compound and a 5-HT1A receptor partial agonist. Ipsapirone (TVX Q 7821) also exhibits 5-HT1A receptor antagonistic effect, and only at high doses it can also produce an inhibitory effect on 5-HT2 and the α1-adrenergic function.	price>
R-R-3384	Iprindole CAS No.5560-72-5	Iprindole/CAS No.5560-72-5, a tricyclic indole antidepressant, is a weak inhibitor of the uptake of noradrenaline and 5-HT.	price>
R-R-3385	cis-(Z)-Flupentixol dihydrochloride CAS No.51529-01-2	cis-(Z)-Flupentixol dihydrochloride/CAS No.51529-01-2 is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively.	price>
R-C-1686	MK 0557 CAS:328232-95-7	MK-0557 is a highly selective,orally administered neuropeptide NPY5R antagonist,could limit weight regain after very-low-calorie diet(VLCD)-induced weight loss.Neuropeptide Y(NPY)is a potent orexigenic neuropeptide,and antagonism of NPY Y1 and NPY Y5 receptors(NPYxR)is considered a potentially important anti-obesity drug target.	price>
R-R-3386	Prucalopride-13C,d3 CAS No.2140306-00-7	Prucalopride-13C,d3/CAS No.2140306-00-7 is the 13C- and deuterium labeled Prucalopride.	price>
R-R-3387	LY 344864 racemate CAS No.186543-64-6	LY 344864 racemate/CAS No.186543-64-6 is a 5-HT1F receptor agonist extracted from patent US 5708187 A.	price>

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