Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3407	LY320135 CAS No.176977-56-3	LY320135/CAS No.176977-56-3 is a potent and selective antagonist of CB1 receptor, with a Ki of 141 nM. LY320135 also binds to 5-HT2 and muscarinic receptors with Kis of 6.4 μM and 2.1 μM, respectively. LY320135 exhibits neuroprotective effect.	price>
R-R-3408	U92016A hydrochloride CAS No.149654-41-1	U92016A hydrochloride/CAS No.149654-41-1 is a potent, metabolically stable, orally acitive 5-HT1A receptor agonist with an exceptionally high degree of intrinsic activity. U92016A hydrochloride binds with high affinity to human 5-HT1A receptors expressed in Chinese hamster ovary cells (Ki=0.2 nM).	price>
R-R-3409	PRX933 hydrochloride CAS No.639029-42-8	PRX933 hydrochloride/CAS No.639029-42-8 is a 5-HT2c receptor agonist extracted from patent WO 2014140631 A1.	price>
R-R-3410	Norfluoxetine-d5 hydrochloride CAS No.1188265-34-0	Norfluoxetine-d5 (hydrochloride)/CAS No.1188265-34-0 is deuterium labeled 3-Phenyl-3-(4-(trifluoromethyl)phenoxy)propan-1-amine hydrochloride.	price>
R-R-3411	Bifeprunox mesylate CAS No.350992-13-1	Bifeprunox mesylate/CAS No.350992-13-1 is a potent dopamine D2-like and 5-HT1A receptor partial agonist with pKis of 7.19 and 8.83 for cortex 5-HT1A and striatum D2, and a pEC50 of 6.37 for hippocampus 5-HT1A, respectively. Bifeprunox mesylate is an antipsychotic for the research of schizophrenia.	price>
R-R-3412	CP-135807 CAS No.151272-90-1	CP-135807/CAS No.151272-90-1 is an orally active and selective 5-HT1D agonist (IC50=3.1 nM), bovine). CP-135807 mediates central psychoactivity and can be used in antidepressant research.	price>
R-R-3413	Vortioxetine-d8 CAS No.2140316-62-5	Vortioxetine-d8/CAS No.2140316-62-5 is a deuterium labeled Vortioxetine. Vortioxetine is an inhibitor of 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT, with Ki values of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.	price>
R-R-3414	Isopteropodine CAS No.5171-37-9	Isopteropodine/CAS No.5171-37-9 is heteroyohimbine-type oxindole alkaloid components of Uncaria tomentosa (Willd.) DC. Isopteropodine acts as positive modulators of muscarinic M1 and 5-HT2 receptors.	price>
R-R-3415	Anpirtoline hydrochloride CAS No.99201-87-3	Anpirtoline hydrochloride/CAS No.99201-87-3 is a hydrochloride of anpirtoline. Anpirtoline is a agonist of 5-HT1B.	price>
R-R-3416	Lurasidone-d8 CAS No.1132654-54-6	Lurasidone-d8/CAS No.1132654-54-6 is deuterium labeled Lurasidone. Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7 with IC50s of 1.68 and 0.495 nM, respectively. Lurasidone (SM-13496) is also a partial agonist of 5-HT1A receptor with an IC50 of 6.75 nM.	price>

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