Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-C-1731	Vorapaxar (MK-5348) CAS: 618385-01-6	Vorapaxar(SCH 530348),an antiplatelet agent,is a selective,orally active,and competitive thrombin receptor protease-activated receptor(PAR-1)antagonist (Ki=8.1nM).Vorapaxar(SCH 530348)inhibits thrombin receptor-activating peptide (TRAP)-induced platelet aggregation in a dose-dependent manner.	price>
R-R-3431	Brexpiprazole-d8-1 CAS No.1427049-19-1	Brexpiprazole-d8-1/CAS No.1427049-19-1 is the deuterium labeled Brexpiprazole[1]. Brexpiprazole (OPC-34712), an atypical orally active antipsychotic agent, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).	price>
R-R-3432	CP 93129 dihydrochloride CAS No.879089-64-2	CP 93129 dihydrochloride/CAS No.879089-64-2 is a potent 5HT1B receptor agonist. CP 93129 dihydrochloride has the potential for parkinson disease research.	price>
R-C-1734	Olopatadine Hydrochlorde CAS:140462-76-6	Olopatadine hydrochloride is a dual acting histamine H1-receptor antagonist and mast cell stabilizer.	price>
R-C-1737	Cloprostenol Sodium CAS:55028-72-3	Cloprostenol sodium salt(ICI 80996 sodium salt)is a potent synthetic prostaglandin analogue,acts as a luteolytic agent,and is a PGF2α receptor agonist.	price>
R-C-1764	PF429242 CAS：947303-87-9	PF 429242 is a reversible,competitive inhibitor of sterol regulatory element-binding protein(SREBP)site 1 protease.	price>
R-C-1765	Treprostinil (LRX-15) CAS：81846-19-7	Treprostinil(LRX-15)is a potent DP1 and EP2 agonist with EC50 values of 0.6±0.1 and 6.2±1.2nM,respectively.	price>
R-C-1766	Pitolisant CAS:362665-56-3	Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor(Ki=0.16nM).	price>
R-C-1770	Amiselimod hydrochloride CAS:942398-84-7	Amiselimod hydrochloride is a novel sphingosine 1-phosphate receptor-1(S1P1) modulator,designed to reduce the bradycardia effects associated with fingolimod and other S1P receptor modulators.	price>
R-C-1771	SB408124 CAS:288150-92-5	SB-408124 is a selective non-peptide orexin OX1 receptor antagonist(Kb values are 21.7 and 1405 nM for human OX1 and OX2 receptors respectively).Blocks orexin-A induced grooming following oral administration in vivo.	price>

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