Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3485	Nemonapride CAS No.75272-39-8	Nemonapride/CAS No.75272-39-8 is a highly potent dopamine D2 receptor antagonist with a Ki of 0.06 nM. Nemonapride also activates 5-HT1A receptor with an IC50 of 34 nM. Nemonapride is an antipsychotic that readily passes through the blood brain barrier and exhibits potent neuroleptic effects in animals.	price>
R-R-3486	ARC 239 CAS No.67339-62-2	ARC 239/CAS No.67339-62-2 is an α2B/C-adrenergic receptor antagonist with pKi of 7.06 and 6.95 for rat kidney α2B and human α2C, respectively. ARC 239 also inhibits 5-HT1A receptor with a Ki of 63.1 nM.	price>
R-R-3487	7-Desmethyl-agomelatine-d3 CAS No.2749427-92-5	7-Desmethyl-agomelatine-d3/CAS No.2749427-92-5 is a deuterium labeled 7-Desmethyl-agomelatine. 7-Desmethyl-agomelatine is a metabolite of Agomelatine.	price>
R-C-1788	TCS OX2 29 CAS：372523-75-6	TCS-OX2-29 is a potent,high affinities and selective orexin-2 receptor(OX2R) antagonist with an IC50 value of 40nM and a pKI value of 7.5.TCS-OX2-29 displays ~250-fold selectivity for OX2 over OX1.	price>
R-R-3488	Vortioxetine-d8 hydrobromide	Vortioxetine-d8 (hydrobromide) is the deuterium labeled Vortioxetine hydrobromide. Vortioxetine hydrobromide is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with Ki values of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.	price>
R-R-3489	LE 300 CAS No.274694-98-3	LE 300/CAS No.274694-98-3 is a potent and selective dopamine D1-like receptor antagonist with Kis of 1.9 nM and 7.5 nM in CHO cell membranes expressing human dopamine D1 and D5 receptors, respectively. LE 300 is an antagonist of the 5-HT2A receptor with a pA2 of 8.32 in a rat tail artery assay.	price>
R-R-3490	Rizatriptan-d6 benzoate CAS No.1216984-85-8	Rizatriptan-d6 (benzoate)/CAS No.1216984-85-8 is the deuterium labeled Rizatriptan benzoate. Rizatriptan benzoate is a 5-HT1 agonist triptan agent for the treatment of migraine headaches.	price>
R-R-3491	5-HT3 antagonist 5 CAS No.901599-43-7	5-HT3 antagonist 5/CAS No.901599-43-7 is a quinoxalin-2-carboxamide compound, a 5-HT3 receptor antagonist. 5-HT3 antagonist 5 exerts antagonism on 5-HT3 agonist and 2-methyl-5-HT, and shows anti-depressant effect in mice.	price>
R-C-1797	SCH58261 CAS：160098-96-4	SCH 58261 is a potent,selective and competitive antagonist of adenosine A2A receptor with an IC50 of 15 nM,and displays 323-,53-and 100-fold more selective for A2A receptor than A1,A2B,and A3 receptors,respectively.	price>
R-R-3512	Namodenoson CAS No.163042-96-4	Namodenoson (CF-102)/CAS No.163042-96-4 is a selective A3 adenosine receptor (A3AR) agonist (Ki=0.33 nM). Namodenoson displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively.	price>

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