Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3310	5-HT1A modulator 1 CAS No.142477-34-7	5-HT1A modulator 1/CAS No.142477-34-7 displays very high affinities for the 5HT1A, adrenergic α1 and dopamine D2 receptor with IC50s of 2 ±0.3 nM, 10 ± 3 nM and 40 ±9 nM, respectively.	price>
R-R-3311	E-3620 CAS No.151213-86-4	E-3620/CAS No.151213-86-4 is a potent 5-HT3 receptor antagonist. E-3620 can be used for the research of dyskinesi and gastrointestinal motility.	price>
R-R-3312	S-14506 hydrochloride CAS No.286369-38-8	S-14506 hydrochloride/CAS No.286369-38-8 is a potent 5-HT1A agonist, as well as 5-HT2A/2C antagonist. S-14506 hydrochloride displays dopamine antagonist properties by blocking dopamine D2 receptors. S-14506 hydrochloride inhibits the in vivo binding of [3H]raclopride in striatum and olfactory bulbs. S-14506 hydrochloride has the potential for the research of anxiolytic agent.	price>
R-R-3313	Amperozide CAS No.75558-90-6	Amperozide/CAS No.75558-90-6 is an atypical antipsychotic that acts as an antagonist of the 5-HT2 receptor with a Ki value of 26 nM. Amperozide has a low affinity for D2 receptors.	price>
R-R-3314	BMY 14802 CAS No.105565-56-8	BMY 14802/CAS No.105565-56-8 is a sigma-1 receptor (σ1R) antagonist, as well as an agonist at serotonin (5-HT) 1A and adrenergic alpha-1 receptors.	price>
R-R-3315	LY 165163 CAS No.1814-64-8	LY 165163/CAS No.1814-64-8 is a potent 5-HT presynaptic receptor agonist. LY 165163 significantly decreases 5-HTP accumulation and increases DOPA accumulation in the cortex and striatum.	price>
R-R-3316	Iferanserin CAS No.58754-46-4	Iferanserin (S-MPEC)/CAS No.58754-46-4 is a selective 5-HT receptor (serotonin receptor) antagonist with an affinity for 5-HT2A receptor. Iferanserin has the potential for internal hemorrhoid disease treatment.	price>
R-R-3317	Olanzapine-d3 CAS No.786686-79-1	Olanzapine-d3/CAS No.786686-79-1 is the deuterium labeled Olanzapine. Olanzapine is a selective, orally active monoaminergic antagonist with high affinity binding to serotonin H1, 5HT2A/2C, 5HT3, 5HT6 (Ki=7, 4, 11, 57, and 5 nM, respectively), dopamine D1-4 (Ki=11 to 31 nM), muscarinic M1-5 (Ki=1.9-25 nM), and adrenergic α1 receptors (Ki=19 nM). Olanzapine is an atypical antipsychotic.	price>
R-R-3318	Keto Ziprasidone CAS No.884305-07-1	Keto Ziprasidone/CAS No.884305-07-1 is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a combined 5-HT (serotonin) and dopamine receptor antagonist.	price>
R-R-3319	(R)-Mirtazapine CAS No.61364-37-2	(R)-Mirtazapine ((R)-Org3770)/CAS No.61364-37-2 is a R(−)-enantiomer of Mirtazapine with antinociceptive properties in an animal model of acute thermal nociception. (R)-Mirtazapine is a 5-HT3 receptor antagonist. (R)-Mirtazapine is mainly metabolized by CYP3A4.	price>

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