Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3314	BMY 14802 CAS No.105565-56-8	BMY 14802/CAS No.105565-56-8 is a sigma-1 receptor (σ1R) antagonist, as well as an agonist at serotonin (5-HT) 1A and adrenergic alpha-1 receptors.	price>
R-R-3315	LY 165163 CAS No.1814-64-8	LY 165163/CAS No.1814-64-8 is a potent 5-HT presynaptic receptor agonist. LY 165163 significantly decreases 5-HTP accumulation and increases DOPA accumulation in the cortex and striatum.	price>
R-R-3316	Iferanserin CAS No.58754-46-4	Iferanserin (S-MPEC)/CAS No.58754-46-4 is a selective 5-HT receptor (serotonin receptor) antagonist with an affinity for 5-HT2A receptor. Iferanserin has the potential for internal hemorrhoid disease treatment.	price>
R-R-3317	Olanzapine-d3 CAS No.786686-79-1	Olanzapine-d3/CAS No.786686-79-1 is the deuterium labeled Olanzapine. Olanzapine is a selective, orally active monoaminergic antagonist with high affinity binding to serotonin H1, 5HT2A/2C, 5HT3, 5HT6 (Ki=7, 4, 11, 57, and 5 nM, respectively), dopamine D1-4 (Ki=11 to 31 nM), muscarinic M1-5 (Ki=1.9-25 nM), and adrenergic α1 receptors (Ki=19 nM). Olanzapine is an atypical antipsychotic.	price>
R-R-3318	Keto Ziprasidone CAS No.884305-07-1	Keto Ziprasidone/CAS No.884305-07-1 is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a combined 5-HT (serotonin) and dopamine receptor antagonist.	price>
R-R-3319	(R)-Mirtazapine CAS No.61364-37-2	(R)-Mirtazapine ((R)-Org3770)/CAS No.61364-37-2 is a R(−)-enantiomer of Mirtazapine with antinociceptive properties in an animal model of acute thermal nociception. (R)-Mirtazapine is a 5-HT3 receptor antagonist. (R)-Mirtazapine is mainly metabolized by CYP3A4.	price>
R-R-3320	OPC-14523 hydrochloride CAS No.145969-31-9	OPC-14523 hydrochloride/CAS No.145969-31-9 is an orally active sigma and 5-HT1A receptor agonist, with high affinity for sigma receptors (σ1/2 IC50=47/56 nM), the 5-HT1A receptor (IC50=2.3 nM), and the 5-HT transporter (IC50=80 nM). OPC-14523 hydrochloride shows antidepressant-like activity.	price>
R-R-3321	Clozapine-d4 CAS No.204395-52-8	Clozapine-d4/CAS No.204395-52-8 is the deuterium labeled Clozapine. Clozapine is an antipsychotic used for the research of schizophrenia. Clozapine has high affinity for a number of neuroreceptors.	price>
R-R-3322	F 13714 fumarate CAS No.208109-39-1	F13714 fumarate/CAS No.208109-39-1, a selective 5-HT1A receptor biased agonist, shows antidepressant-like properties after a single administration in the mouse model of chronic mild stress.	price>
R-R-3323	CJ033466 CAS No.519148-48-2	CJ033466/CAS No.519148-48-2 is a novel and selective 5-HT4 receptor partial agonist with an EC50 of 9 nM and has gastroprokinetic effect.	price>

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