Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-C-1604	Conivaptan hydrochloride CAS:168626-94-6	Conivaptan(hydrochloride)is a non-peptide antagonist of vasopressin receptor, with Ki values of 0.48 and 3.04 nM for rat liver V1A receptor and rat kidney V2 receptor respectively.	price>
R-R-3304	Cyamemazine CAS No.3546-03-0	Cyamemazine/CAS No.3546-03-0 is a neuroleptic agent that contains the phenothiazine chromophore. Cyamemazine is often used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki of 12 nM), 5-HT2A (Ki = 1.5 nM) and 5-HT2C (Ki of 75 nM) receptors antagonist with antipsychotic activity.	price>
R-C-1605	Lixivaptan CAS：168079-32-1	Lixivaptan(VPA-985,WAY-VPA985)is an orally active and selective vasopressin receptor V2 antagonist,with IC50 values of 1.2 and 2.3 nM for human and rat V2,respectively.	price>
R-R-3305	Quetiapine hemifumarate (Standard) CAS No.111974-72-2	Quetiapine (hemifumarate) (Standard)/CAS No.111974-72-2 is the analytical standard of Quetiapine (hemifumarate). This product is intended for research and analytical applications. Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor. Quetiapine hemifumarate has moderate to high affinity for the human D2, HT1A, 5-HT2A, 5-HT2C receptor with pKis of 7.25, 5.74, 7.54, 5.55. Antidepressant and anxiolytic effects.	price>
R-R-3306	Eltoprazine hydrochloride CAS No.98206-09-8	Eltoprazine (DU 28853) hydrochloride/CAS No.98206-09-8 is a 5-HT1A/5-HT1B receptors agonist and a 5-HT2C receptor antagonist. Eltoprazine hydrochloride shows antiaggressive and anxiogenic effects.	price>
R-R-3307	Eplivanserin hemifumarate CAS No.130580-02-8	Eplivanserin (SR-46349) hemifumarate/CAS No.130580-02-8 is a potent, selective and orally active 5-HT2A receptor antagonist, with an IC50 of 5.8 nM in rat cortical membrane, and a Kd of 1.14 nM. Eplivanserin hemifumarate displays >20-fold selectivity more selective for 5-HT2A than 5-HT2B and 5-HT2C.	price>
R-R-3308	4F 4PP oxalate CAS No.144734-36-1	4F 4PP (oxalate)/CAS No.144734-36-1 is a selective 5-HT2A antagonist with almost as high affinity (Ki= 5.3 nM) as ketanserin but with a much lower affinity for 5-HT2C sites (Ki= 620 nM).	price>
R-R-3309	PNU-142633 CAS No.187665-65-2	PNU-142633/CAS No.187665-65-2 is a high affinity, selective and orally active 5-HT1D receptor agonist with Kis of 6 nM and > 18 000 nM for human 5-HT1D receptor and human 5-HT1B receptor, respectively. PNU-142633 has anti-migraine efficacy.	price>
R-R-3310	5-HT1A modulator 1 CAS No.142477-34-7	5-HT1A modulator 1/CAS No.142477-34-7 displays very high affinities for the 5HT1A, adrenergic α1 and dopamine D2 receptor with IC50s of 2 ±0.3 nM, 10 ± 3 nM and 40 ±9 nM, respectively.	price>
R-R-3311	E-3620 CAS No.151213-86-4	E-3620/CAS No.151213-86-4 is a potent 5-HT3 receptor antagonist. E-3620 can be used for the research of dyskinesi and gastrointestinal motility.	price>

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