Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3262	WAY-100135 dihydrochloride CAS No.149055-79-8	WAY-100135 dihydrochloride/CAS No.149055-79-8 is a selective antagonist at presynaptic and postsynaptic 5-HT1A receptor, with an IC50 of 34 nM at the rat hippocampal 5-HT1A receptor. WAY-100135 dihydrochloride has potential antipsychotic properties.	price>
R-R-3263	7-Desmethyl-agomelatine CAS No.152302-45-9	7-Desmethyl-agomelatine/CAS No.152302-45-9 is a metabolite of Agomelatine. Agomelatineis a potent agonist at melatonin receptors (MT1 and MT2), and also is an antagonist of 5-HT2C.	price>
R-R-3264	Donitriptan CAS No.170912-52-4	Donitriptan/CAS No.170912-52-4 is a potent, high efficacy agonist at 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively.	price>
R-C-1565	Relugolix (TAK-385) CAS：737789-87-6	Relugolix(RVT-601,TAK-385)is a selective antagonist of the gonadotropin-releasing hormone receptor(GnRHR)with IC50 of 0.33 nM and 0.32 nM for human GnRHR and monkey GnRHR,respectively.	price>
R-R-3265	Strictosidinic acid CAS No.150148-81-5	Strictosidinic acid/CAS No.150148-81-5, an orally active glycoside indole monoterpene alkaloid isolated from Psychotria myriantha leaves, inhibits precursor enzymes of 5-HT biosynthesis and reduces the 5-HT levels. Strictosidinic acid has peripheral analgesic and antipyretic activities in mice.	price>
R-R-3266	Felcisetrag CAS No.916075-84-8	Felcisetrag (TD-8954)/CAS No.916075-84-8 is an orally active, potent and selective 5-HT4 receptor agonist with gastrointestinal prokinetic properties. Felcisetrag has high affinity (pKi =9.4) for human 5-HT4(c) receptors.	price>
R-R-3267	Pirenperone CAS No.75444-65-4	Pirenperone (R 47465)/CAS No.75444-65-4 is a 5-HT2 serotonin receptor antagonist. Pirenperone exhibits modest anxiolytic activity.	price>
R-R-3268	GR 55562 dihydrochloride CAS No.159533-25-2	GR 55562 (dihydrochloride)/CAS No.159533-25-2 is a selective 5-HT1B receptor antagonist. GR 55562 can be used for the research of nerve disease.	price>
R-R-3269	Perospirone hydrochloride CAS No.129273-38-7	Perospirone hydrochloride (SM-9018)/CAS No.129273-38-7 is an orally active antagonist of 5-HT2A receptor (Ki of 0.6 nM) and dopamine D2 receptor (Ki of 1.4 nM). Perospirone hydrochloride is also a partial agonist of 5-HT1A receptor (Ki of 2.9 nM). Perospirone hydrochloride is an atypical antipsychotic agent and has the potential for schizophrenic disease research.	price>
R-R-3270	Urapidil CAS No.34661-75-1	Urapidil/CAS No.34661-75-1 is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist.	price>

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