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Catalog name Description price
R-C-2804 Eglumegad (LY354740) CAS:176199-48-7 Eglumegad(LY354740)is a highly potent and selective group II(mGlu2/3)receptor agonist with IC50s of 5 and 24nM on transfected human mGlu2 and mGlu3 receptors,respectively. price>
R-C-2805 NKP608 CAS:177707-12-9 NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective,specific and potent antagonist at the neurokinin-1(NK-1)receptor both in vitro(IC50=2.6nM)and in vivo. price>
R-C-2806 Sumanirole maleate CAS:179386-44-8 Sumanirole maleate(U-95666E;PNU-95666E)is a highly selective D2 receptor full agonist with an ED50 of about 46nM.Sumanirole was developed for the treatment of Parkinson is disease and restless leg syndrome. price>
R-C-2809 LY 344864 CAS:186544-26-3 LY344864 is a selective receptor agonist with an affinity of 6 nM(Ki)at the recently cloned 5-HT1F receptor. price>
R-C-2811 NGB 2904 CAS:189060-98-8 NGB 2904 is an orally active and selective dopamine(DA)D3 receptor antagonist.NGB 2904 can be used for the research of cocaine addiction. price>
R-C-2814 LY 379268 CAS:191471-52-0 LY379268 is a potent,selective and brain-penetrant mGlu2/3R agonist with EC50 values of 2.69nM(mGlu2)and 4.48nM(mGlu3).LY379268 has no activity on human mGlu 1a,4a,5a or 7a receptors.LY379268 has antioxidant and neuroprotective effects. price>
R-C-2965 SB-269970 SB269970 is a potent and selective 5-HT7 receptor antagonist. price>
R-C-2967 Olcegepant CAS：204697-65-4 Olcegepant also known as BIBN-4096 or BIBN-4096BS is is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1)receptor. price>
R-C-2968 SB271046 CAS：209481-20-9 SB271046 is a potent,selective and orally active 5-HT6 receptor antagonist with pKi of 8.9,exhibits 200-fold greater selectivity over other 5-HT receptor subtypes. price>
R-C-2969 SB269652 CAS：215802-15-6 SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor(D2R).SB269652 binds in a bitopic manner at one protomer of a D2R dimer and modulates the binding of dopamine at a second protomer. price>