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Catalog name Description price
R-R-4403 Dopamine D2 receptor agonist-3 CAS No.1257326-24-1 Dopamine D2 receptor agonist-3 (compound 3)/CAS No.1257326-24-1 is a selective D2 receptor partial agonist and Dopamine D3 receptor antagonist (with pEC50 of 8.3 and <5.5 respectively). price>
R-R-4404 Ropinirole-d7 hydrochloride CAS No.1261396-31-9 Ropinirole-d7 (hydrochloride)/CAS No.1261396-31-9 is the deuterium labeled Ropinirole hydrochloride[1]. Ropinirole (SKF 101468) hydrochloride is an orally active, potent D3/D2 receptor agonist with a Ki of 29 nM for D2 receptor. Ropinirole hydrochloride has pEC50s of 7.4, 8.4 and 6.8 for hD2, hD3 and hD4 receptors, respectively. Ropinirole hydrochloride has no affinity for the D1 receptors. price>
R-R-4405 (E/Z)-Chlorprothixene-d6 hydrochloride CAS No.1246832-91-6 (E/Z)-Chlorprothixene-d6 hydrochloride/CAS No.1246832-91-6 is the deuterium labeled (E/Z)-Chlorprothixene hydrochloride. price>
R-R-4406 Fluphenazine-d8 dihydrochloride Fluphenazine-d8 (dihydrochloride) is the deuterium labeled Fluphenazine dihydrochloride. Fluphenazine dihydrochloride is a phenothiazine-class D1DR and D2DR inhibitor; used to deliver Fluphenazine to biological systems in studies probing the effects and metabolic fates of this commonly used dopamine antagonist. price>
R-R-4407 Bromperidol hydrochloride CAS No.59453-24-6 Bromperidol (R-11333) hydrochloride/CAS No.59453-24-6 possesses antipsychotic activity, with a high affinity for central dopamine receptors D2. Bromperidol hydrochloride can kill Mycobacteria in a synergistic manner with Spectinomycin. price>
R-R-4408 PG01037 dihydrochloride CAS No.675599-62-9 PG01037 (dihydrochloride)/CAS No.675599-62-9 is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM. price>
R-R-4409 Cabergoline-d6 CAS No.2738376-76-4 Cabergoline-d6 is deuterium labeled Cabergoline. Cabergoline is an ergot derived-dopamine D2-like receptor agonist that has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively). price>
R-R-4410 OS-3-106 CAS No.1580000-17-4 OS-3-106/CAS No.1580000-17-4 is a potent, BBB-penetrated and selective dopamine D3 receptor (D3R) agonist. OS-3-106 binds with high affinity (Ki = 0.2 nM) at the D3R. OS-3-106 can be used for psychoactivator addiction research. price>
R-R-4411 Clomipramine-d3 hydrochloride CAS No.1398065-86-5 Clomipramine-d3 (hydrochloride)/CAS No.1398065-86-5 is a deuterium labeled Clomipramine hydrochloride. Clomipramine hydrochloride is a serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) blocker with Ki of 0.14, 54 and 3 nM, respectively. price>
R-R-4412 Fluphenazine-d8 CAS No.1323633-98-2 Fluphenazine-d8/CAS No.1323633-98-2 is the deuterium labeled Fluphenazine. Fluphenazine is a potent, orally active phenothiazine-based dopamine receptor antagonist. Fluphenazine blocks neuronal voltage-gated sodium channels. Fluphenazine acts primarily through antagonism of postsynaptic dopamine-2 receptors in mesolimbic, nigrostriatal, and tuberoinfundibular neural pathways. Fluphenazine can antagonize Methylphenidate-induced stereotyped gnawing and inhibit climbing behaviour in mice. Fluphenazine can be used for researching psychosis and painful peripheral neuropathy associated with diabetes and has potential to inhibit SARS-CoV-2. price>