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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4406 Fluphenazine-d8 dihydrochloride Fluphenazine-d8 (dihydrochloride) is the deuterium labeled Fluphenazine dihydrochloride. Fluphenazine dihydrochloride is a phenothiazine-class D1DR and D2DR inhibitor; used to deliver Fluphenazine to biological systems in studies probing the effects and metabolic fates of this commonly used dopamine antagonist. price>
R-R-4407 Bromperidol hydrochloride CAS No.59453-24-6 Bromperidol (R-11333) hydrochloride/CAS No.59453-24-6 possesses antipsychotic activity, with a high affinity for central dopamine receptors D2. Bromperidol hydrochloride can kill Mycobacteria in a synergistic manner with Spectinomycin. price>
R-R-4408 PG01037 dihydrochloride CAS No.675599-62-9 PG01037 (dihydrochloride)/CAS No.675599-62-9 is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM. price>
R-R-4409 Cabergoline-d6 CAS No.2738376-76-4 Cabergoline-d6 is deuterium labeled Cabergoline. Cabergoline is an ergot derived-dopamine D2-like receptor agonist that has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively). price>
R-R-4410 OS-3-106 CAS No.1580000-17-4 OS-3-106/CAS No.1580000-17-4 is a potent, BBB-penetrated and selective dopamine D3 receptor (D3R) agonist. OS-3-106 binds with high affinity (Ki = 0.2 nM) at the D3R. OS-3-106 can be used for psychoactivator addiction research. price>
R-R-4411 Clomipramine-d3 hydrochloride CAS No.1398065-86-5 Clomipramine-d3 (hydrochloride)/CAS No.1398065-86-5 is a deuterium labeled Clomipramine hydrochloride. Clomipramine hydrochloride is a serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) blocker with Ki of 0.14, 54 and 3 nM, respectively. price>
R-R-4412 Fluphenazine-d8 CAS No.1323633-98-2 Fluphenazine-d8/CAS No.1323633-98-2 is the deuterium labeled Fluphenazine. Fluphenazine is a potent, orally active phenothiazine-based dopamine receptor antagonist. Fluphenazine blocks neuronal voltage-gated sodium channels. Fluphenazine acts primarily through antagonism of postsynaptic dopamine-2 receptors in mesolimbic, nigrostriatal, and tuberoinfundibular neural pathways. Fluphenazine can antagonize Methylphenidate-induced stereotyped gnawing and inhibit climbing behaviour in mice. Fluphenazine can be used for researching psychosis and painful peripheral neuropathy associated with diabetes and has potential to inhibit SARS-CoV-2. price>
R-R-4413 Sonepiprazole CAS No.170858-33-0 Sonepiprazole (PNU-101387G)/CAS No.170858-33-0 is a selective D4 dopamine antagonist with Kis of 3.6, 10.1, 5147, and 7430 nM for rD4-Dopamine, hD4.2-Dopamine, rD2-Dopamine, and Histamine-H1 receptors, respectively. price>
R-R-4414 Haloperidol-d4-1 CAS No.136765-35-0 Haloperidol-d4-1/CAS No.136765-35-0 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. price>
R-R-4415 Dexpramipexole-d3 dihydrochloride CAS No.1432230-09-5 Dexpramipexole-d3 (dihydrochloride)/CAS No.1432230-09-5 is the deuterium labeled Dexpramipexole. Dexpramipexole((R)-Pramipexole), also known as R-(+)-Pramipexole, is a neuroprotective agent and weak non-ergoline dopamine agonist. price>