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Catalog name Description price
R-R-4393 FAUC 213 CAS No.337972-47-1 FAUC 213/CAS No.337972-47-1 is an orally active and highly selective dopamine D4 receptor complete antagonist with a Ki of 2.2 nM for hD4.4. FAUC 213 has less activity on D2 and D3 receptors (Kis of 3.4 μM, 5.3 μM for hD2, hD3, respectively). FAUC 213 can cross the blood-brain barrier (BBB). FAUC 213 exhibits atypical antipsychotic characteristic. price>
R-R-4394 BP 897 hydrochloride CAS No.314776-92-6 BP 897 hydrochloride/CAS No.314776-92-6 is a potent and partial dopamine D3 receptor agonist and a weak D2 receptor antagonist. BP 897 hydrochloride displays a high affinity at the dopamine D3 receptor (Ki=0.92 nM) and a 70 times lower affinity at the D2 receptor (Ki=61 nM). price>
R-R-4395 FAUC 346 CAS No.474432-65-0 FAUC 346/CAS No.474432-65-0, a highly selective D3 partial agonist (EC50 = 1.5 nM). price>
R-R-4396 Bromperidol (Standard) CAS No.10457-90-6 Bromperidol (Standard)/CAS No.10457-90-6 is the analytical standard of Bromperidol. This product is intended for research and analytical applications. Bromperidol (R-11333) possesses antipsychotic activity, with a high affinity for central dopamine receptors D2. Bromperidol can kill Mycobacteria in a synergistic manner with Spectinomycin. price>
R-R-4397 L-DOPA-13C CAS No.586971-29-1 L-DOPA-13C/CAS No.586971-29-1 is the 13C labeled L-DOPA[1]. L-DOPA (Levodopa) is an orally active metabolic precursor of neurotransmitters dopamine. L-DOPA can cross the blood-brain barrier and is converted into dopamine in the brain. price>
R-R-4398 Asimilobine CAS No.6871-21-2 Asimilobine/CAS No.6871-21-2 is an aporphine isoquinoline alkaloid isolated from plant species of Magnolia obobata Thun. Asimilobine is a dopamine biosynthesis inhibitor and a serotonergic receptor antagonist. Asimilobine shows an antimalarial and anti-cancer activity. price>
R-R-4399 PNU-177864 CAS No.250266-51-4 PNU-177864/CAS No.250266-51-4 is a potent, selective and orally active dopamine D3 receptor antagonist. PNU-177864 is structurally consistent with a cationic amphiphilic agent (CAD) and induces phospholipidosis in vivo. PNU-177864 antischizophrenic activity. price>
R-R-4400 NPEC-caged-dopamine CAS No.1257326-23-0 NPEC-caged-dopamine/CAS No.1257326-23-0 is a caged version of dopamine. NPEC-caged-Dopamine was used by applying focal photolysis with UV light (360 nm) to releases dopamine, which leads to D1 receptor activation. price>
R-R-4401 Timiperone CAS No.57648-21-2 Timiperone/CAS No.57648-21-2 has a strong affinity for cerebral dopamine D2 receptor. Timiperone has antipsychotic activity, and inhibits stereotyped behaviour. Timiperone can be used for research of schizophrenia. price>
R-R-4402 Pramipexole-d5 dihydrochloride CAS No.1217601-58-5 Pramipexole-d5 (dihydrochloride)/CAS No.1217601-58-5 is deuterium labeled Pramipexole (dihydrochloride). Pramipexole dihydrochloride is a selective and blood-brain barrier (BBB) penetrant dopamine D2-type receptor agonist, with Kis of 2.2 nM, 3.9 nM, 0.5 nM and 1.3 nM for D2-type receptor, D2, D3 and D4 receptors, respectively. price>