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Catalog name Description price
R-R-4386 PD 168568 dihydrochloride CAS No.1782532-06-2 PD 168568 dihydrochloride/CAS No.1782532-06-2 is a orally active and potent dopamine receptor D4 (DRD4) antagonist. PD 168568 dihydrochloride contains an isoindolinone and is selective for the D4 receptor versus D2 and D3, with Ki values of 8.8, 1842, and 2682 nM, respectively. PD 168568 dihydrochloride can be used for glioblastoma (GBM) research. price>
R-R-4387 Amisulpride-d5 CAS No.1216626-17-3 Amisulpride-d5/CAS No.1216626-17-3 is the deuterium labeled Amisulpride. Amisulpride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively. price>
R-R-4388 Cabergoline-d5 CAS No.1426173-20-7 Cabergoline-d5/CAS No.1426173-20-7 is the deuterium labeled Cabergoline. Cabergoline is an ergot derived-dopamine D2-like receptor agonist that has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively). price>
R-R-4389 FAUC 365 CAS No.474432-66-1 FAUC 365/CAS No.474432-66-1 is a highly dopamine D3 receptor-selective antagonist with Ki values of 0.5 nM, 340, 2600, and 3600 nM at D3, D4.4, D2short, and D2Long receptors, respectively. FAUC 365 can be used for the research of schizophrenia, and Parkinson disease. price>
R-R-4390 SK609 hydrochloride CAS No.1092797-77-7 SK609 hydrochloride/CAS No.1092797-77-7 is a dopamine D3 receptor (D3R) selective agonist with an EC50 of 1109 nM. SK609 hydrochloride has the potential for parkinson research. price>
R-R-4391 Levosulpiride-d3 CAS No.124020-27-5 Levosulpiride-d3/CAS No.124020-27-5 is the deuterium labeled Levosulpiride. Levosulpiride (RV-12309) is the (S)-enantiomer of sulpiride, which is a D2 receptor a antagonist, an atypical antipsychotic agent of the benzamide class. price>
R-R-4392 CP 226269 CAS No.220941-93-5 CP 226269/CAS No.220941-93-5 is a potent dopamine D4 receptor agonist that induces calcium flux with EC50 of 32.0 nM. CP 226269 can be used in the research of schizophrenia and other related diseases. price>
R-R-4393 FAUC 213 CAS No.337972-47-1 FAUC 213/CAS No.337972-47-1 is an orally active and highly selective dopamine D4 receptor complete antagonist with a Ki of 2.2 nM for hD4.4. FAUC 213 has less activity on D2 and D3 receptors (Kis of 3.4 μM, 5.3 μM for hD2, hD3, respectively). FAUC 213 can cross the blood-brain barrier (BBB). FAUC 213 exhibits atypical antipsychotic characteristic. price>
R-R-4394 BP 897 hydrochloride CAS No.314776-92-6 BP 897 hydrochloride/CAS No.314776-92-6 is a potent and partial dopamine D3 receptor agonist and a weak D2 receptor antagonist. BP 897 hydrochloride displays a high affinity at the dopamine D3 receptor (Ki=0.92 nM) and a 70 times lower affinity at the D2 receptor (Ki=61 nM). price>
R-R-4395 FAUC 346 CAS No.474432-65-0 FAUC 346/CAS No.474432-65-0, a highly selective D3 partial agonist (EC50 = 1.5 nM). price>