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Catalog name Description price
R-C-2776 Ebrotidine CAS:100981-43-9 Ebrotidine(FI 3542)is a competitive H2-receptor antagonist(Ki=27.5nM)with a potent antisecretory activity and evidenced gastroprotection. price>
R-C-2777 CY 208-243 CAS：100999-26-6 CY 208-243 is a drug which acts as a dopamine agonist selective for the D1subtype.Unlike most D1-selective agonists,it shows efficacy in animal models of Parkinson is disease. price>
R-C-2780 Otenzepad (AF-DX 116) CAS：102394-31-0 Otenzepad(AF-DX 116)is a selective and competitive M2 muscarinic acetylcholine receptor antagonist,with IC50 values of 640nM and 386nM for rabbit peripheral lung and rat heart,respectively. price>
R-C-2781 VUF 10460 CAS：1028327-66-3 VUF10460 is a non-imidazole histamine H4 receptor agonist;binds to rat H4 receptor with a pKi of 7.46. price>
R-C-2792 TCN 238 CAS:125404-04-8 TCN238 is an orally bioavailable mGlu4 receptor positive allosteric modulator (PAM)with an EC50 of 1μM. price>
R-C-2797 L-732,138 CAS:148451-96-1 L-732138 is a selective,potent and competitive neurokinin-1(NK-1)receptor antagonist with an IC50 of 2.3nM.L-732138 has 200-fold more potent in cloned human NK-1 receptors than cloned rat NK-1 receptors,and has>1000-fold more potent than human NK-2 and NK-3 receptors.L-732138 can reduce hyperalgesia and has antitumor action. price>
R-C-2800 GR 103691 CAS:162408-66-4 GR 103691 is a potent,selective dopamine D3 receptor antagonist with a Ki value of 0.4nM.GR 103691 shows more than 100-fold selectivity for human dopamine human(h)D3 over hD4 and hD1 sites. price>
R-C-2804 Eglumegad (LY354740) CAS:176199-48-7 Eglumegad(LY354740)is a highly potent and selective group II(mGlu2/3)receptor agonist with IC50s of 5 and 24nM on transfected human mGlu2 and mGlu3 receptors,respectively. price>
R-C-2805 NKP608 CAS:177707-12-9 NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective,specific and potent antagonist at the neurokinin-1(NK-1)receptor both in vitro(IC50=2.6nM)and in vivo. price>
R-C-2806 Sumanirole maleate CAS:179386-44-8 Sumanirole maleate(U-95666E;PNU-95666E)is a highly selective D2 receptor full agonist with an ED50 of about 46nM.Sumanirole was developed for the treatment of Parkinson is disease and restless leg syndrome. price>