Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-2763	O-Phospho-L-serine-13C3,15N CAS No.2734706-69-3	O-Phospho-L-serine-13C3,15N/CAS No.2734706-69-3 is the 13C- and 15N-labeled O-Phospho-L-serine. O-Phospho-L-serine is the immediate precursor to L-serine in the serine synthesis pathway, and an agonist at the group III mGluR receptors (mGluR4, mGluR6, mGluR7, and mGluR8); O-Phospho-L-serine also acts as a weak antagonist for mGluR1 and a potent antagonist for mGluR2.	price>
R-R-2764	(S)-4CPG CAS No.134052-73-6	(S)-4CPG ((S)-4-Carboxyphenylglycine)/CAS No.134052-73-6 is a potent mGluR2 agonist. (S)-4CPG reduces hyperalgesia and allodynia associated with sciatic nerve contraction injury in rats. (S)-4CPG can be used in research on neurological diseases.	price>
R-R-2765	CBiPES CAS No.353235-01-5	CBiPES/CAS No.353235-01-5 is a potent mGlu2 positive allosteric modulator with an EC50 value of 92.8 nM. CBiPES attenuates stress-induced hyperthermia and Phencyclidine-induced hyperlocomotor activity. CBiPES can be used for research of neurological diseases.	price>
R-R-2766	SIB-1757 CAS No.31993-01-8	SIB-1757/CAS No.31993-01-8 is a highly selective and noncompetitive antagonist of mGlu5 receptor with an IC50 of 0.4 μM.	price>
R-R-2767	L-Glutamine-13C5,15N2,d5 CAS No.2123439-02-9	L-Glutamine-13C5,15N2,d5/CAS No.2123439-02-9 is the deuterium, 13C-, and 15-labeled L-Glutamine. L-Glutamine (L-Glutamic acid 5-amide) is a non-essential amino acid present abundantly throughout the body and involved in many metabolic processes. L-Glutamine provides a source of carbons for oxidation in some cells.	price>
R-R-2768	CBiPES hydrochloride CAS No.856702-40-4	CBiPES hydrochloride/CAS No.856702-40-4 is a mGlu2 receptor positive allosteric modulator (EC50: 92.8 nM). CBiPES hydrochloride attenuates stress-induced hyperthermia and PCP-induced hyperlocomotor activity. CBiPES hydrochloride can be used for research of neurological disease.	price>
R-C-1069	REVERSINE CAS：656820-32-5	Reversine is a potent human A3 adenosine receptor antagonist with Ki of 0.66 μM, and a pan-aurora A/B/C kinase inhibitor with IC50 of 12 nM/13 nM/20 nM,respectively.Also used for stem cell dedifferentiation.	price>
R-R-2769	(S,S)-BMS-984923 CAS No.1375752-77-4	(S,S)-BMS-984923/CAS No.1375752-77-4 is a less active (S,S)-enantiomer of BMS-984923. (S,S)-BMS-984923 shows an EC50 >1μM for mGluR5 receptor. BMS-984923 is a potent mGluR5 silent allosteric modulator. (S,S)-BMS-984923 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-R-2770	ML289 CAS No.1382481-79-9	ML289 (VU0463597)/CAS No.1382481-79-9 is a potent, selective, and CNS-penetrant mGlu3 (IC50=0.66 μM) negative allosteric modulator. ML289 displays >15-fold selectivity over mGlu2 and is inactive against mGlu5. ML289 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-R-2771	VU0469650 CAS No.1443748-47-7	VU0469650/CAS No.1443748-47-7 is a potent, selective and CNS-penetrated negative allosteric modulator of mGlu1 receptor, with an IC50 of 99 nM.	price>

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