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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4337 SKF 83959 hydrobromide CAS No.67287-95-0 SKF83959 hydrobromide/CAS No.67287-95-0 is a potent and selective dopamine D1-like receptor partial agonist. SKF83959 hydrobromide Ki values for rat D1, D5, D2 and D3 receptors are 1.18, 7.56, 920 and 399 nM, respectively. SKF83959 hydrobromide is a potent allosteric modulator of sigma (σ)-1 receptor. SKF83959 hydrobromide belongs to benzazepine family and has improvements on cognitive dysfunction. price>
R-R-4338 PF-06256142 CAS No.1609583-14-3 PF-06256142/CAS No.1609583-14-3 is a potent, selective, CNS-penetrant and orally active agonist of the D1 receptor, with an EC50 and Ki of 33 nM and 12 nM, respectively. price>
R-R-4339 Tavapadon CAS No.1643489-24-0 Tavapadon (PF-06649751)/CAS No.1643489-24-0 is an orally active and highly selective dopamine D1/D5 receptor partial agonist. price>
R-R-4340 Mesdopetam hemitartrate CAS No.2562346-14-7 Mesdopetam (IRL790) hemitartrate/CAS No.2562346-14-7 is a dopamine D3 receptor antagonist (Ki=90 nM; IC50=9.8 μM for human recombinant D3 receptor) with psychomotor stabilizing properties. Mesdopetam hemitartrate is used for the research of motor and psychiatric complications in Parkinson disease. price>
R-R-4341 Dopamine D2 receptor antagonist-1 CAS No.1055411-77-2 Dopamine D2 receptor antagonist-1/CAS No.1055411-77-2 is a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R) with sub-mM affinity. price>
R-R-4342 Propionylpromazine hydrochloride CAS No.7681-67-6 Propionylpromazine hydrochloride (Propiopromazine hydrochloride)/CAS No.7681-67-6, a dopamine receptor D2 (DRD2) antagonist, can be used in the research of Parkinson disease. price>
R-R-4343 Quinelorane dihydrochloride CAS No.97548-97-5 Quinelorane dihydrochloride (LY163502)/CAS No.97548-97-5 is a potent dopamine D3/D2 receptor agonist. Quinelorane has the potential for neurological and psychiatric disorders research. price>
R-R-4344 (Rac)-PF-06256142 CAS No.1609580-97-3 (Rac)-PF-06256142/CAS No.1609580-97-3 is the less effective enantiomer of PF-06256142 (HY-119943). (Rac)-PF-06256142 is an agonist of D1 receptor, with an EC50 of 107 nM. price>
R-R-4345 Carmoxirole hydrochloride CAS No.115092-85-8 Carmoxirole hydrochloride (EMD 45609 hydrochloride)/CAS No.115092-85-8 is a selective, peripherally acting dopamine D2 receptor agonist and exhibits antihypertensive activities in vivo. price>
R-R-4346 Acetophenazine dimaleate CAS No.5714-00-1 Acetophenazine dimaleate/CAS No.5714-00-1, a phenothiazine derivative, is an antipsychotic agent. Acetophenazine dimaleate primarily blocks dopamine D2 receptors in the brain. Acetophenazine dimaleate can be used for researching psychotic disorders such as schizophrenia and anxious depression. price>