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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4354 Molindone hydrochloride CAS No.15622-65-8 Molindone hydrochloride (EN-1733A)/CAS No.15622-65-8 is a therapeutic antipsychotic, used in the treatment of schizophrenia, works by blocking the effects of dopamine in the brain, leading to diminished psychoses. price>
R-R-4355 ABT-724 trihydrochloride CAS No.587870-77-7 ABT-724 trihydrochloride/CAS No.587870-77-7 is a potent and highly selective dopamine D4 receptor agonist with an EC50 of 12.4 nM for human dopamine D4 receptor. ABT-724 trihydrochloride is a potent partial agonist at the rat D4 (EC50 of 14.3 nM) and the ferret D4 receptor (EC50 of 23.2 nM), and has no effect on dopamine D1, D2, D3, or D5 receptors. ABT-724 trihydrochloride could be useful for the treatment of erectile dysfunction and has favorable side-effect profile. price>
R-R-4356 Bacopaside X CAS No.94443-88-6 Bacopaside X/CAS No.94443-88-6 is found in Bacopa monnieri, and shows a binding affinity toward the D1 receptor. price>
R-R-4357 Naxagolide CAS No.88058-88-2 Naxagolide ((+)-PHNO; Dopazinol)/CAS No.88058-88-2 is a potent dopamine D2 (Dopamine Receptor) agonist. Naxagolide has the potential for the research of parkinson disease (PD). price>
R-R-4358 JNJ-37822681 dihydrochloride CAS No.2108806-02-4 JNJ-37822681 dihydrochloride/CAS No.2108806-02-4 is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. price>
R-R-4359 (Rac)-Razpipadon CAS No.1643462-93-4 PW0464/CAS No.1643462-93-4, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP). price>
R-R-4360 MIF-1 TFA CAS No.35240-69-8 MIF-1 TFA (Melanostatin)/CAS No.35240-69-8, an endogenous brain peptide, is a potent dopamine receptor allosteric modulator. MIF-1 TFA inhibits melanin formation. MIF-1 TFA blocks the effects of opioid receptor activation to modulate the analgesic effects. MIF-1 TFA accesses from the blood to the CNS by directly crossing the blood-brain barrier (BBB). price>
R-R-4361 Alizapride hydrochloride CAS No.59338-87-3 Alizapride/CAS No.59338-87-3 is a potent antiemetic, acting as a dopamine receptor antagonist. Alizapride also used in human digestive disorders. price>
R-R-4362 Aramisulpride CAS No.71675-90-6 Aramisulpride/CAS No.71675-90-6 is a dopamine D2 receptor and serotonin receptor antagonist used for the research of metabolic disorders. price>
R-R-4363 (R)-Preclamol hydrochloride CAS No.89874-80-6 (R)-Preclamol hydrochloride ((+)-3-PPP hydrochloride)/CAS No.89874-80-6 is the R-enantiomer of Preclamol hydrochloride. (R)-Preclamol hydrochloride is a DA agonist with autoreceptor as well as postsynaptic receptor stimulatory properties. price>