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Catalog name Description price
R-R-4304 Ralmitaront CAS No.2133417-13-5 Ralmitaront (RO6889450)/CAS No.2133417-13-5 is an orally active agonist of trace amine-associated receptor 1 (TAAR1) with a EC50 value of 110.4 nM. Ralmitaront has antipsychotic, cognitively improvement, and antidepressant activity in rodents. Ralmitaront can be used as a neurosuppressant in the study of neuro-related diseases, such as schizophrenia (SCZ), schizoaffective disorder. price>
R-R-4305 Ropinirole hydrochloride CAS No.91374-20-8 Ropinirole (SKF 101468) hydrochloride/CAS No.91374-20-8 is an orally active, potent D3/D2 receptor agonist with a Ki of 29 nM for D2 receptor. Ropinirole hydrochloride has pEC50s of 7.4, 8.4 and 6.8 for hD2, hD3 and hD4 receptors, respectively. Ropinirole hydrochloride has no affinity for the D1 receptors. price>
R-R-4306 Pramipexole dihydrochloride CAS No.104632-25-9 Pramipexole dihydrochloride/CAS No.104632-25-9 is a selective and blood-brain barrier (BBB) penetrant dopamine D2-type receptor agonist, with Kis of 2.2 nM, 3.9 nM, 0.5 nM and 1.3 nM for D2-type receptor, D2, D3 and D4 receptors, respectively. price>
R-R-4307 Lisuride maleate CAS No.19875-60-6 Lisuride (maleate)/CAS No.19875-60-6 is a potent agonist of dopamine with a probably direct action on dopaminergic receptors. Lisuride (maleate) is an ergot derivative. Lisuride (maleate) releases the premenstrual mastalgia without significant side effects. price>
R-R-4308 L-741626 CAS No.81226-60-0 L-741626/CAS No.81226-60-0 is a selective D2 dopamine receptor antagonist, with the Ki values of 2.4, 100 and 220 nM for human D2, D3 and D4 receptors respectively. price>
R-R-4309 3-O-Methyldopa CAS No.300-48-1 3-O-Methyldopa (3-Methoxy-L-tyrosine)/CAS No.300-48-1 is a metabolite of L-DOPA which is formed by catechol-O-methyltransferase (COMT). 3-O-Methyldopa competitively inhibits the pharmacodynamics of l-DOPA and dopamine. price>
R-R-4310 Droperidol CAS No.548-73-2 Droperidol/CAS No.548-73-2 is a butyrophenone-type Dopamine-2 receptor antagonist. price>
R-R-4311 Loxapine succinate CAS No.27833-64-3 Loxapine succinate/CAS No.27833-64-3 is an orally active dopamine inhibitor, 5-HT receptor antagonist and also a dibenzoxazepine anti-psychotic agent. Loxapine can also suppresses bacterial efflux pump activity and inhibit intracellular multiple-antibiotic-resistant Salmonella enterica serovar Typhimurium in macrophages. price>
R-R-4312 Nomifensine CAS No.24526-64-5 Nomifensine/CAS No.24526-64-5 is a norepinephrine-dopamine reuptake inhibitor, increases the amount of synaptic norepinephrine and dopamine available to receptors by blocking the dopamine and norepinephrine reuptake transporters. price>
R-R-4313 A68930 hydrochloride CAS No.130465-39-3 A68930 hydrochloride/CAS No.130465-39-3, as a dopamine D1 receptor agonist, can be used for the research of bronchiectasis. price>