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Catalog name Description price
R-R-4298 Raclopride CAS No.84225-95-6 Raclopride/CAS No.84225-95-6 is a dopamine D2/D3 receptor antagonist with potential antipsychotic effects. Raclopride binds to D2 and D3 receptors with Kis of 1.8 nM and 3.5 nM, respectively. price>
R-R-4299 SKF-82958 hydrobromide CAS No.74115-01-8 SKF-82958 ((±)-SKF 82958) hydrobromide/CAS No.74115-01-8 is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM). price>
R-R-4300 Dihydrexidine hydrochloride CAS No.137417-08-4 Dihydrexidine hydrochloride (DAR-0100 hydrochloride)/CAS No.137417-08-4 is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist, with an IC50 of 10 nM for D1 receptor. Dihydrexidine hydrochloride exhibits potent antiparkinsonian activity. Dihydrexidine hydrochloride can stimulate YAP phosphorylation. price>
R-R-4301 Tetrahydropalmatine CAS No.2934-97-6 Tetrahydropalmatine/CAS No.2934-97-6 possesses analgesic effects. Tetrahydropalmatine acts through inhibition of amygdaloid release of dopamine to inhibit an epileptic attack in rats. price>
R-R-4302 Pergolide mesylate CAS No.66104-23-2 Pergolide mesylate (Pergolide methanesulfonate)/CAS No.66104-23-2, an Ergoline derivative, is a potent and orally active dopamine D1 and D2 receptors agonist. price>
R-R-4303 Tetrahydroberberine CAS No.522-97-4 Tetrahydroberberine/CAS No.522-97-4 is a different kind of living thing that can be extended and divided into parts. Tetrahydroberberine is a kind of effective D2 receptor antagonistic force. Tetrahydroberberine has the ability to strengthen the stomach and relieve the pressure on the stomach. price>
R-R-4304 Ralmitaront CAS No.2133417-13-5 Ralmitaront (RO6889450)/CAS No.2133417-13-5 is an orally active agonist of trace amine-associated receptor 1 (TAAR1) with a EC50 value of 110.4 nM. Ralmitaront has antipsychotic, cognitively improvement, and antidepressant activity in rodents. Ralmitaront can be used as a neurosuppressant in the study of neuro-related diseases, such as schizophrenia (SCZ), schizoaffective disorder. price>
R-R-4305 Ropinirole hydrochloride CAS No.91374-20-8 Ropinirole (SKF 101468) hydrochloride/CAS No.91374-20-8 is an orally active, potent D3/D2 receptor agonist with a Ki of 29 nM for D2 receptor. Ropinirole hydrochloride has pEC50s of 7.4, 8.4 and 6.8 for hD2, hD3 and hD4 receptors, respectively. Ropinirole hydrochloride has no affinity for the D1 receptors. price>
R-R-4306 Pramipexole dihydrochloride CAS No.104632-25-9 Pramipexole dihydrochloride/CAS No.104632-25-9 is a selective and blood-brain barrier (BBB) penetrant dopamine D2-type receptor agonist, with Kis of 2.2 nM, 3.9 nM, 0.5 nM and 1.3 nM for D2-type receptor, D2, D3 and D4 receptors, respectively. price>
R-R-4307 Lisuride maleate CAS No.19875-60-6 Lisuride (maleate)/CAS No.19875-60-6 is a potent agonist of dopamine with a probably direct action on dopaminergic receptors. Lisuride (maleate) is an ergot derivative. Lisuride (maleate) releases the premenstrual mastalgia without significant side effects. price>