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Catalog name Description price
R-R-4294 Cabergoline CAS No.81409-90-7 Cabergoline/CAS No.81409-90-7 is an ergot derived-dopamine D2-like receptor agonist that has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively). price>
R-R-4295 Fluphenazine dihydrochloride CAS No.146-56-5 Fluphenazine dihydrochloride/CAS No.146-56-5 is a potent, orally active phenothiazine-based dopamine receptor antagonist. Fluphenazine dihydrochloride blocks neuronal voltage-gated sodium channels. Fluphenazine dihydrochloride acts primarily through antagonism of postsynaptic dopamine-2 receptors in mesolimbic, nigrostriatal, and tuberoinfundibular neural pathways. Fluphenazine dihydrochloride can antagonize Methylphenidate-induced stereotyped gnawing and inhibit climbing behaviour in mice. Fluphenazine dihydrochloride can be used for researching psychosis and painful peripheral neuropathy associated with diabetes and has potential to inhibit SARS-CoV-2. price>
R-R-4296 ONC206 CAS No.1638178-87-6 ONC206/CAS No.1638178-87-6 is an analogue of TRAIL inducer ONC201. ONC206 is a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations. ONC206 has broad-spectrum anti-tumor activity. price>
R-R-4297 Sulpiride CAS No.15676-16-1 Sulpiride/CAS No.15676-16-1 is an orally active dopamine D2/D3 receptor antagonist. Sulpiride is an atypical antipsychotic agent of the benzamide family. Sulpiride can be used in research into anxiety, depression and breast cancer. price>
R-R-4298 Raclopride CAS No.84225-95-6 Raclopride/CAS No.84225-95-6 is a dopamine D2/D3 receptor antagonist with potential antipsychotic effects. Raclopride binds to D2 and D3 receptors with Kis of 1.8 nM and 3.5 nM, respectively. price>
R-R-4299 SKF-82958 hydrobromide CAS No.74115-01-8 SKF-82958 ((±)-SKF 82958) hydrobromide/CAS No.74115-01-8 is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM). price>
R-R-4300 Dihydrexidine hydrochloride CAS No.137417-08-4 Dihydrexidine hydrochloride (DAR-0100 hydrochloride)/CAS No.137417-08-4 is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist, with an IC50 of 10 nM for D1 receptor. Dihydrexidine hydrochloride exhibits potent antiparkinsonian activity. Dihydrexidine hydrochloride can stimulate YAP phosphorylation. price>
R-R-4301 Tetrahydropalmatine CAS No.2934-97-6 Tetrahydropalmatine/CAS No.2934-97-6 possesses analgesic effects. Tetrahydropalmatine acts through inhibition of amygdaloid release of dopamine to inhibit an epileptic attack in rats. price>
R-R-4302 Pergolide mesylate CAS No.66104-23-2 Pergolide mesylate (Pergolide methanesulfonate)/CAS No.66104-23-2, an Ergoline derivative, is a potent and orally active dopamine D1 and D2 receptors agonist. price>
R-R-4303 Tetrahydroberberine CAS No.522-97-4 Tetrahydroberberine/CAS No.522-97-4 is a different kind of living thing that can be extended and divided into parts. Tetrahydroberberine is a kind of effective D2 receptor antagonistic force. Tetrahydroberberine has the ability to strengthen the stomach and relieve the pressure on the stomach. price>