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Catalog name Description price
R-R-4289 SKF 81297 CAS No.71636-61-8 SKF 81297/CAS No.71636-61-8 is a potent and selective dopamine D1 receptor agonist. price>
R-R-4290 Fallypride CAS No.166173-78-0 Fallypride/CAS No.166173-78-0 is a potent antagonist of dopamine D2/D3 receptor. Fallypride, in the form of fallypride (18F), can be used as a positron emission tomography (PET) radiotracer. price>
R-C-2591 GRI 977143 CAS:325850-81-5 GRI977143 is a selective lysophosphatidic acid 2(LPA2)receptor non-lipid agonist (EC50=3.3μM).GRI977143 does not activate other LPA GPCRs at concentrations up to 10μM. price>
R-R-4291 Octoclothepin maleate salt CAS No.4789-68-8 Octoclothepin maleate salt/CAS No.4789-68-8, an orally active neuroleptic agent, is a dual SR-2A and D2DR inhibitor. Octoclothepin maleate salt reveals an intensive central depressant action in a series of observational and instrumental procedures in rodents. price>
R-R-4292 Clozapine N-oxide dihydrochloride CAS No.2250025-93-3 Clozapine N-oxide dihydrochloride/CAS No.2250025-93-3 is a major metabolite of Clozapine and a human muscarinic designer receptors (DREADDs) agonist. Clozapine N-oxide dihydrochloride activates the DREADD receptor hM3Dq and hM4Di. Clozapine N-oxide dihydrochloride can cross the blood-brain barrier. Clozapine is a potent dopamine antagonist and also a potent and selective muscarinic M4 receptor (EC50=11 nM) agonist. price>
R-R-4293 SKF 38393 hydrochloride CAS No.62717-42-4 SKF 38393 hydrochloride/CAS No.62717-42-4 is a selective agonist of the dopamine D1 receptor (D1DR) with an IC50 of 110 nM. price>
R-R-4294 Cabergoline CAS No.81409-90-7 Cabergoline/CAS No.81409-90-7 is an ergot derived-dopamine D2-like receptor agonist that has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively). price>
R-R-4295 Fluphenazine dihydrochloride CAS No.146-56-5 Fluphenazine dihydrochloride/CAS No.146-56-5 is a potent, orally active phenothiazine-based dopamine receptor antagonist. Fluphenazine dihydrochloride blocks neuronal voltage-gated sodium channels. Fluphenazine dihydrochloride acts primarily through antagonism of postsynaptic dopamine-2 receptors in mesolimbic, nigrostriatal, and tuberoinfundibular neural pathways. Fluphenazine dihydrochloride can antagonize Methylphenidate-induced stereotyped gnawing and inhibit climbing behaviour in mice. Fluphenazine dihydrochloride can be used for researching psychosis and painful peripheral neuropathy associated with diabetes and has potential to inhibit SARS-CoV-2. price>
R-R-4296 ONC206 CAS No.1638178-87-6 ONC206/CAS No.1638178-87-6 is an analogue of TRAIL inducer ONC201. ONC206 is a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations. ONC206 has broad-spectrum anti-tumor activity. price>
R-R-4297 Sulpiride CAS No.15676-16-1 Sulpiride/CAS No.15676-16-1 is an orally active dopamine D2/D3 receptor antagonist. Sulpiride is an atypical antipsychotic agent of the benzamide family. Sulpiride can be used in research into anxiety, depression and breast cancer. price>