Products classification
ABOUT US
Email:
sales@ruixibiotech.com
Tel.:
02988811435
Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4275 (R,R)-CXCR2-IN-2 CAS No.1838123-22-0 (R,R)-CXCR2-IN-2/CAS No.1838123-22-0, diastereoisomer of CXCR2-IN-2 (compound 68), is a brain penetrant CXCR2 antagonist with a pIC50 of 9 and 6.8 in the Tango assay and d in the HWB Gro-α induced CD11b expression assay, respectively. price>
R-R-4276 MSX-127 CAS No.6616-56-4 MSX-127/CAS No.6616-56-4 is a CXCR4 antagonist. MSX-127 inhibits cancer metastasis. price>
R-R-4277 MSX-130 CAS No.4051-59-6 MSX-130/CAS No.4051-59-6 is a CXCR4 antagonist. MSX-130 inhibits cancer metastasis. price>
R-R-4278 Vimnerixin CAS No.1418112-77-2 Vimnerixin (AZD4721)/CAS No.1418112-77-2 is the potent and orally active antagonist of acidic CXC chemokine receptor 2 (CXCR2). Vimnerixin has the potential for the research of inflammatory disease. price>
R-R-4279 AZD8309 CAS No.333742-48-6 AZD8309 is an orally active antagonist of CXCR2. AZD8309 has the ability to regulate the transmigration of neutrophils. AZD8309 can be used in the study of inflammatory diseases. price>
R-R-4280 ACT-660602 CAS No.1646267-59-5 ACT-660602/CAS No.1646267-59-5 is an orally active antagonist of chemokine receptor (CXCR3) with an IC50 value of 204 nM. ACT-660602 inhibits T-cell migration and shows efficacy in acute lung ingury model. ACT-660602 can be used for autoimmune diseases research. price>
R-R-4281 SCH 563705 CAS No.473728-58-4 SCH 563705/CAS No.473728-58-4 is a potent and orally available CXCR2 and CXCR1 antagonist, with IC50s of 1.3 nM, 7.3 nM and Kis of 1 and 3 nM, respectively. price>
R-R-4282 CTCE-0214 CAS No.577782-52-6 CTCE-0214/CAS No.577782-52-6 is a chemokine CXC receptor 4 (CXCR4) agonist, SDF-1α (stromal cell-derived factor-1α) peptide analog. CTCE-0214 shows anti-inflammatory activity, and can be used in inflammation sepsis and systemic inflammatory syndromes research. price>
R-R-4283 SRT3109 CAS No.1204707-71-0 SRT3109/CAS No.1204707-71-0 is an antagonist of CXCR2, with a pIC50 of 8.2, and used in the research of chemokine mediated diseases. price>
R-R-4284 Plerixafor-d4 CAS No.1246819-87-3 Plerixafor-d4/CAS No.1246819-87-3 is the deuterium labeled Plerixafor. Plerixafor (AMD 3100) is a selective CXCR4 antagonist with an IC50 of 44 nM. Plerixafor, an immunostimulant and a hematopoietic stem cell (HSC) mobilizer, is an allosteric agonist of CXCR7. Plerixafor inhibits HIV-1 and HIV-2 replication with an EC50 of 1-10 nM. price>