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Catalog name Description price
R-C-2535 Ambrisentan（BSF208075，LU208075） CAS No. 177036-94-1 Ambrisentan(LU-208075,BSF-208075)is a highly selective antagonist of the endothelin-1 type A receptor,used in the treatment of pulmonary arterial hypertension(PAH). price>
R-R-4235 AMG 487 CAS No.473719-41-4 AMG 487/CAS No.473719-41-4 is an orally active and selective antagonist of CXC chemokine receptor 3 (CXCR3) which inhibits the binding of CXCL10 and CXCL11 to CXCR3 with IC50s of 8.0 and 8.2 nM, respectively. price>
R-C-2536 Canagliflozin hemihydrate CAS：928672-86-0 Canagliflozin hemihydrate(JNJ28431754 hemihydrate) is a selective SGLT2 inhibitor with IC50s of 2nM,3.7nM,and 4.4nM for mSGLT2, rSGLT2,and hSGLT2 in CHOK cells,respectively. price>
R-R-4236 Reparixin CAS No.266359-83-5 Reparixin/CAS No.266359-83-5 is a non-competitive allosteric inhibitor of the chemokine receptors CXCR1 and CXCR2 activation with IC50s of 1 and 100 nM, respectively. price>
R-C-2537 Ipragliflozin (ASP1941) CAS：761423-87-4 Ipragliflozin(ASP1941)is an orally active and selective SGLT2 inhibitor with IC50s of 7.38 and 1876nM,6.73 and 1166nM,5.64 and 1380nM for human SGLT2 and SGLT1,rat SGLT2 and SGLT1,mouse SGLT2 and SGLT1,respectively.Antidiabetic agent. price>
R-R-4237 Plerixafor octahydrochloride CAS No.155148-31-5 Plerixafor octahydrochloride (AMD3100 octahydrochloride)/CAS No.155148-31-5 is a selective CXCR4 antagonist with an IC50 of 44 nM. price>
R-C-2538 Tofogliflozin(CSG 452) CAS：1201913-82-7 Tofogliflozin(CSG-452)is a potent and highly specific sodium/glucose cotransporter 2(SGLT2)inhibitor with Ki values of 2.9,14.9,and 6.4nM for human, rat,and mouse SGLT2. price>
R-R-4238 Navarixin CAS No.473727-83-2 Navarixin (SCH 527123)/CAS No.473727-83-2 is a CXCR1 and CXCR2 antagonist that is potent, allosteric, and orally active, with Kd values of 41 nM for cynomolgus CXCR1 and 0.20 nM, 0.20 nM, 0.08 nM for mouse, rat and cynomolgus monkey CXCR2, respectively. price>
R-C-2539 Plerixafor（ AMD310） CAS：110078-46-1 Plerixafor(AMD 3100)is a selective CXCR4 antagonist with an IC50 of 44nM.Plerixafor,an immunostimulant and a hematopoietic stem cell(HSC)mobilizer, is an allosteric agonist of CXCR7.Plerixafor inhibits HIV-1 and HIV-2 replication with an EC50 of 1-10nM. price>
R-R-4239 AZD-5069 CAS No.878385-84-3 AZD-5069/CAS No.878385-84-3 is a potent CXCR2 chemokine receptor antagonist, used for caner treatment. price>