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Catalog name Description price
R-C-2533 Canagliflozin (JNJ 28431754) CAS：842133-18-0 Canagliflozin(JNJ 28431754)is a selective SGLT2 inhibitor with IC50s of 2nM, 3.7nM,and 4.4nM for mSGLT2,rSGLT2,and hSGLT2 in CHOK cells,respectively. price>
R-R-4233 (Rac)-Sograzepide CAS No.168161-71-5 (Rac)-Sograzepide/CAS No.168161-71-5 is an antagonist of cholecystokinin B (CCK-B) receptor, and has the potential of reducing the secretion of gastric acid. price>
R-R-4234 CCK antagonist 1 CAS No.742116-45-6 CCK antagonist 1 (compound 3d)/CAS No.742116-45-6 is a CCK antagonist with IC50s of 1.1 μM and 4 μM for CCK1 and CCK2, respectively. CCK antagonist 1 can be used for research of cancer and mental disease. price>
R-C-2535 Ambrisentan（BSF208075，LU208075） CAS No. 177036-94-1 Ambrisentan(LU-208075,BSF-208075)is a highly selective antagonist of the endothelin-1 type A receptor,used in the treatment of pulmonary arterial hypertension(PAH). price>
R-R-4235 AMG 487 CAS No.473719-41-4 AMG 487/CAS No.473719-41-4 is an orally active and selective antagonist of CXC chemokine receptor 3 (CXCR3) which inhibits the binding of CXCL10 and CXCL11 to CXCR3 with IC50s of 8.0 and 8.2 nM, respectively. price>
R-C-2536 Canagliflozin hemihydrate CAS：928672-86-0 Canagliflozin hemihydrate(JNJ28431754 hemihydrate) is a selective SGLT2 inhibitor with IC50s of 2nM,3.7nM,and 4.4nM for mSGLT2, rSGLT2,and hSGLT2 in CHOK cells,respectively. price>
R-R-4236 Reparixin CAS No.266359-83-5 Reparixin/CAS No.266359-83-5 is a non-competitive allosteric inhibitor of the chemokine receptors CXCR1 and CXCR2 activation with IC50s of 1 and 100 nM, respectively. price>
R-C-2537 Ipragliflozin (ASP1941) CAS：761423-87-4 Ipragliflozin(ASP1941)is an orally active and selective SGLT2 inhibitor with IC50s of 7.38 and 1876nM,6.73 and 1166nM,5.64 and 1380nM for human SGLT2 and SGLT1,rat SGLT2 and SGLT1,mouse SGLT2 and SGLT1,respectively.Antidiabetic agent. price>
R-R-4237 Plerixafor octahydrochloride CAS No.155148-31-5 Plerixafor octahydrochloride (AMD3100 octahydrochloride)/CAS No.155148-31-5 is a selective CXCR4 antagonist with an IC50 of 44 nM. price>
R-C-2538 Tofogliflozin(CSG 452) CAS：1201913-82-7 Tofogliflozin(CSG-452)is a potent and highly specific sodium/glucose cotransporter 2(SGLT2)inhibitor with Ki values of 2.9,14.9,and 6.4nM for human, rat,and mouse SGLT2. price>