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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4227 A71623 CAS No.130408-77-4 A71623/CAS No.130408-77-4, a CCK-4-based peptide, is a potent and highly selective CCK-A full agonist. The IC50s for A-71623 are 3.7 nM in guinea pig pancreas (CCK-A) and 4500 nM in cerebral cortex (CCK-B) in radioligand binding assays, respectively. price>
R-C-2528 Losartan potassium CAS：124750-99-8 Losartan potassium(DuP-753 potassium)is an angiotensin II receptor type 1 (AT1)antagonist,competing with the binding of angiotensin II to AT1 with an IC50 of 20nM. price>
R-R-4228 Lorglumide sodium salt CAS No.1021868-76-7 Lorglumide sodium salt (CR-1409 sodium salt)/CAS No.1021868-76-7 is a potent cholecystokinin (CCK) receptor antagonist. price>
R-R-4229 Lintitript CAS No.136381-85-6 Lintitript (SR 27897)/CAS No.136381-85-6 is a highly potent, selective, orally active, competitive and non-peptide cholecystokinin (CCK1) receptor antagonist with an EC50 of 6 nM and a Ki of 0.2 nM. Lintitript displays > 33-fold selectivity more selective for CCK1 than CCK2 receptors (EC50 value of 200 nM). Lintitript increases plasma concentration of leptin and food intake as well as plasma concentration of insulin. price>
R-R-4230 Dexloxiglumide CAS No.119817-90-2 Dexloxiglumide/CAS No.119817-90-2 is a selective cholecystokinin type A (CCKA) receptor antagonist. Dexloxiglumide, the active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). price>
R-R-4231 CCK-B Receptor Antagonist 2 CAS No.155412-88-7 CCK-B Receptor Antagonist 2/CAS No.155412-88-7, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82 μM. price>
R-R-4232 L-365260 hemihydrate L-365260 hemihydrate is an orally active and selective antagonist of non-peptide gastrin and brain cholecystokinin receptor (CCK-B), with Kis of 1.9 nM and 2.0 nM, respectively. L-365260 hemihydrate interacts in a stereoselective and competitive manner with guinea pig stomach gastrin and brain CCK receptors. price>
R-C-2533 Canagliflozin (JNJ 28431754) CAS：842133-18-0 Canagliflozin(JNJ 28431754)is a selective SGLT2 inhibitor with IC50s of 2nM, 3.7nM,and 4.4nM for mSGLT2,rSGLT2,and hSGLT2 in CHOK cells,respectively. price>
R-R-4233 (Rac)-Sograzepide CAS No.168161-71-5 (Rac)-Sograzepide/CAS No.168161-71-5 is an antagonist of cholecystokinin B (CCK-B) receptor, and has the potential of reducing the secretion of gastric acid. price>
R-R-4234 CCK antagonist 1 CAS No.742116-45-6 CCK antagonist 1 (compound 3d)/CAS No.742116-45-6 is a CCK antagonist with IC50s of 1.1 μM and 4 μM for CCK1 and CCK2, respectively. CCK antagonist 1 can be used for research of cancer and mental disease. price>