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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4079 2-Arachidonoylglycerol CAS No.53847-30-6 2-Arachidonoylglycerol/CAS No.53847-30-6 is a second endogenous cannabinoid ligand in the central nervous system. price>
R-R-4080 JD-5037 CAS No.1392116-14-1 JD-5037/CAS No.1392116-14-1 is a potent CB1R antagonist with an IC50 of 1.5 nM. price>
R-R-4081 GW405833 hydrochloride CAS No.1202865-22-2 GW405833 hydrochloride/CAS No.1202865-22-2 is a potent and selective cannabinoid-2 (CB2) receptor agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%). GW405833 hydrochloride produces potent antihyperalgesic effects in several rodent models of pain. price>
R-R-4082 Taranabant CAS No.701977-09-5 Taranabant/CAS No.701977-09-5 is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. price>
R-R-4083 Pregnenolone monosulfate sodium CAS No.1852-38-6 Pregnenolone monosulfate sodium (3β-Hydroxy-5-pregnen-20-one monosulfate sodium)/CAS No.1852-38-6 is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of tetrahydrocannabinol (THC) that are mediated by the CB1 receptors. Pregnenolone monosulfate sodium can protect the brain from cannabis intoxication. Pregnenolone monosulfate sodium is also a TRPM3 channel activator, and also can weakly activate TRPM1 channels. price>
R-R-4084 Olorinab CAS No.1268881-20-4 Olorinab (APD 371)/CAS No.1268881-20-4 is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist, with an EC50 of 6.2 nM for hCB2. price>
R-R-4085 Yangonin CAS No.500-62-9 Yangonin/CAS No.500-62-9 exhibits affinity for the human recombinant cannabinoid CB1 receptor with an IC50 and a Ki of 1.79 μM and 0.72 μM, respectively. price>
R-R-4086 AM281 CAS No.202463-68-1 AM281/CAS No.202463-68-1 is a selective CB1 receptor antagonist with an IC50 of 9.91 nM. AM281 inhibits CB2 receptor with an IC50 of 13000 nM. price>
R-R-4087 LY2828360 CAS No.1231220-79-3 LY2828360/CAS No.1231220-79-3 is a slowly acting but efficacious G protein-biased cannabinoid (CB2) agonist, inhibiting cAMP accumulation and activating ERK1/2 signaling. price>
R-R-4088 Monlunabant CAS No.2712480-46-9 Monlunabant ((S)-MRI-1891)/CAS No.2712480-46-9 is a solid dispersions compound, as well as a cannabinoid CB1 receptor inhibitor. price>