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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4084 Olorinab CAS No.1268881-20-4 Olorinab (APD 371)/CAS No.1268881-20-4 is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist, with an EC50 of 6.2 nM for hCB2. price>
R-R-4085 Yangonin CAS No.500-62-9 Yangonin/CAS No.500-62-9 exhibits affinity for the human recombinant cannabinoid CB1 receptor with an IC50 and a Ki of 1.79 μM and 0.72 μM, respectively. price>
R-R-4086 AM281 CAS No.202463-68-1 AM281/CAS No.202463-68-1 is a selective CB1 receptor antagonist with an IC50 of 9.91 nM. AM281 inhibits CB2 receptor with an IC50 of 13000 nM. price>
R-R-4087 LY2828360 CAS No.1231220-79-3 LY2828360/CAS No.1231220-79-3 is a slowly acting but efficacious G protein-biased cannabinoid (CB2) agonist, inhibiting cAMP accumulation and activating ERK1/2 signaling. price>
R-R-4088 Monlunabant CAS No.2712480-46-9 Monlunabant ((S)-MRI-1891)/CAS No.2712480-46-9 is a solid dispersions compound, as well as a cannabinoid CB1 receptor inhibitor. price>
R-R-4089 (±)-Ibipinabant CAS No.362519-49-1 (±)-Ibipinabant ((±)-SLV319)/CAS No.362519-49-1 is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. price>
R-R-4090 CB1 antagonist 4 CAS No.1253641-65-4 CB1 antagonist 4 (compound 8)/CAS No.1253641-65-4 is a peripheral selective cannabinoid receptor type 1 (CB1) receptor antagonist. CB1 antagonist 4 shows limited penetrance to the brain in order to minimize or prevent CNS adverse reactions, and preserves potential antiobesity effects. CB1 antagonist 4 reduces propensity for psychiatric side effects. price>
R-R-4091 Org 27569 CAS No.868273-06-7 Org 27569/CAS No.868273-06-7 is a potent CB1 receptor allosteric modulator, which increases agonist binding, yet blocks agonist-induced CB1 signaling. price>
R-R-4092 GW-405833 CAS No.180002-83-9 GW-405833 (L768242)/CAS No.180002-83-9 is a potent, selective cannabinoid receptor 2 (CB2) agonist with an EC50 of 50.7 nM. GW-405833 also behaves as a noncompetitive CB1 antagonist. GW-405833 suppresses inflammatory and neuropathic pain. price>
R-R-4093 Leelamine hydrochloride CAS No.16496-99-4 Leelamine hydrochloride/CAS No.16496-99-4 is a tricyclic diterpene molecule that is extracted from the bark of pine trees. Leelamine hydrochloride is a cannabinoid receptor type 1 (CB1) agonist and a inhibitor of SREBP1-regulated fatty acid/lipid synthesis in prostate cancer cells that is not affected by androgen receptor status. Leelamine hydrochloride suppresses transcriptional activity of androgen receptor, which is known to regulate fatty acid synthesis[2,3]. price>