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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4073 Fulimetibant CAS No.2231142-90-6 Fulimetibant/CAS No.2231142-90-6 is a bradykinin receptor antagonist. price>
R-R-4074 ELN-441958 CAS No.913064-47-8 ELN-441958/CAS No.913064-47-8 is a potent, neutral, competitive and selective bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor. ELN-441958 has high oral bioavailability, and has low CNS exposure in the mouse. price>
R-R-4075 Bradykinin (2-9) CAS No.16875-11-9 Bradykinin (2-9)/CAS No.16875-11-9 is an amino-truncated Bradykinin peptide. Bradykinin (2-9) is a metabolite of Bradykinin, cleaved by Aminopeptidase P. price>
R-R-4076 Bradykinin (1-5) CAS No.23815-89-6 Bradykinin (1-5)/CAS No.23815-89-6 is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE). price>
R-R-4077 [Hyp3]-Bradykinin CAS No.37642-65-2 [Hyp3]-Bradykinin/CAS No.37642-65-2, naturally occurring peptide hormone, is a bradykinin receptor agonist. [Hyp3]-Bradykinin interacts with B2-bradykinin receptors and stimulates inositol phosphate production in cultured human fibroblasts. price>
R-R-4078 Rimonabant Hydrochloride CAS No.158681-13-1 Rimonabant Hydrochloride (SR 141716A Hydrochloride)/CAS No.158681-13-1 is a highly potent and selective central cannabinoid receptor (CB1) antagonist with an Ki of 1.8 nM. Rimonabant Hydrochloride (SR 141716A Hydrochloride) also inhibits Mycobacterial membrane protein Large 3 (MMPL3). price>
R-R-4079 2-Arachidonoylglycerol CAS No.53847-30-6 2-Arachidonoylglycerol/CAS No.53847-30-6 is a second endogenous cannabinoid ligand in the central nervous system. price>
R-R-4080 JD-5037 CAS No.1392116-14-1 JD-5037/CAS No.1392116-14-1 is a potent CB1R antagonist with an IC50 of 1.5 nM. price>
R-R-4081 GW405833 hydrochloride CAS No.1202865-22-2 GW405833 hydrochloride/CAS No.1202865-22-2 is a potent and selective cannabinoid-2 (CB2) receptor agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%). GW405833 hydrochloride produces potent antihyperalgesic effects in several rodent models of pain. price>
R-R-4082 Taranabant CAS No.701977-09-5 Taranabant/CAS No.701977-09-5 is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. price>