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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4074 ELN-441958 CAS No.913064-47-8 ELN-441958/CAS No.913064-47-8 is a potent, neutral, competitive and selective bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor. ELN-441958 has high oral bioavailability, and has low CNS exposure in the mouse. price>
R-R-4075 Bradykinin (2-9) CAS No.16875-11-9 Bradykinin (2-9)/CAS No.16875-11-9 is an amino-truncated Bradykinin peptide. Bradykinin (2-9) is a metabolite of Bradykinin, cleaved by Aminopeptidase P. price>
R-R-4076 Bradykinin (1-5) CAS No.23815-89-6 Bradykinin (1-5)/CAS No.23815-89-6 is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE). price>
R-R-4077 [Hyp3]-Bradykinin CAS No.37642-65-2 [Hyp3]-Bradykinin/CAS No.37642-65-2, naturally occurring peptide hormone, is a bradykinin receptor agonist. [Hyp3]-Bradykinin interacts with B2-bradykinin receptors and stimulates inositol phosphate production in cultured human fibroblasts. price>
R-R-4078 Rimonabant Hydrochloride CAS No.158681-13-1 Rimonabant Hydrochloride (SR 141716A Hydrochloride)/CAS No.158681-13-1 is a highly potent and selective central cannabinoid receptor (CB1) antagonist with an Ki of 1.8 nM. Rimonabant Hydrochloride (SR 141716A Hydrochloride) also inhibits Mycobacterial membrane protein Large 3 (MMPL3). price>
R-R-4079 2-Arachidonoylglycerol CAS No.53847-30-6 2-Arachidonoylglycerol/CAS No.53847-30-6 is a second endogenous cannabinoid ligand in the central nervous system. price>
R-R-4080 JD-5037 CAS No.1392116-14-1 JD-5037/CAS No.1392116-14-1 is a potent CB1R antagonist with an IC50 of 1.5 nM. price>
R-R-4081 GW405833 hydrochloride CAS No.1202865-22-2 GW405833 hydrochloride/CAS No.1202865-22-2 is a potent and selective cannabinoid-2 (CB2) receptor agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%). GW405833 hydrochloride produces potent antihyperalgesic effects in several rodent models of pain. price>
R-R-4082 Taranabant CAS No.701977-09-5 Taranabant/CAS No.701977-09-5 is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. price>
R-R-4083 Pregnenolone monosulfate sodium CAS No.1852-38-6 Pregnenolone monosulfate sodium (3β-Hydroxy-5-pregnen-20-one monosulfate sodium)/CAS No.1852-38-6 is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of tetrahydrocannabinol (THC) that are mediated by the CB1 receptors. Pregnenolone monosulfate sodium can protect the brain from cannabis intoxication. Pregnenolone monosulfate sodium is also a TRPM3 channel activator, and also can weakly activate TRPM1 channels. price>