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Catalog name Description price
R-R-4069 Icatibant acetate CAS No.138614-30-9 Icatibant acetate (HOE-140 acetate)/CAS No.138614-30-9 is a potent and specific peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively. price>
R-R-4070 Lobradimil CAS No.159768-75-9 Lobradimil (RMP 7)/CAS No.159768-75-9, a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). Lobradimil increases the permeability of the BBB. Lobradimil can be used in the research of brain tumors. price>
R-R-4071 R715 CAS No.185052-09-9 R715/CAS No.185052-09-9 is a selective bradykinin B1 receptor antagonist. R715 significantly attenuates the hyperalgesic effect developed in Streptozotocin(HY-13753)-diabetic mice. price>
R-R-4072 MEN 11270 CAS No.235082-52-7 MEN 11270/CAS No.235082-52-7, a cyclic decapeptide, is a B2 kinin receptor antagonist. MEN 11270 bound with high-affinity to the B2 kinin receptor constitutively expressed by WI38 human fibroblasts, inhibiting 3H-bradykinin (BK) with a pKi value of 10.3. price>
R-R-4073 Fulimetibant CAS No.2231142-90-6 Fulimetibant/CAS No.2231142-90-6 is a bradykinin receptor antagonist. price>
R-R-4074 ELN-441958 CAS No.913064-47-8 ELN-441958/CAS No.913064-47-8 is a potent, neutral, competitive and selective bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor. ELN-441958 has high oral bioavailability, and has low CNS exposure in the mouse. price>
R-R-4075 Bradykinin (2-9) CAS No.16875-11-9 Bradykinin (2-9)/CAS No.16875-11-9 is an amino-truncated Bradykinin peptide. Bradykinin (2-9) is a metabolite of Bradykinin, cleaved by Aminopeptidase P. price>
R-R-4076 Bradykinin (1-5) CAS No.23815-89-6 Bradykinin (1-5)/CAS No.23815-89-6 is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE). price>
R-R-4077 [Hyp3]-Bradykinin CAS No.37642-65-2 [Hyp3]-Bradykinin/CAS No.37642-65-2, naturally occurring peptide hormone, is a bradykinin receptor agonist. [Hyp3]-Bradykinin interacts with B2-bradykinin receptors and stimulates inositol phosphate production in cultured human fibroblasts. price>
R-R-4078 Rimonabant Hydrochloride CAS No.158681-13-1 Rimonabant Hydrochloride (SR 141716A Hydrochloride)/CAS No.158681-13-1 is a highly potent and selective central cannabinoid receptor (CB1) antagonist with an Ki of 1.8 nM. Rimonabant Hydrochloride (SR 141716A Hydrochloride) also inhibits Mycobacterial membrane protein Large 3 (MMPL3). price>