Catalog |
name |
Description |
price |
R-R-4069 |
Icatibant acetate CAS No.138614-30-9 |
Icatibant acetate (HOE-140 acetate)/CAS No.138614-30-9 is a potent and specific peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively. |
price> |
R-R-4070 |
Lobradimil CAS No.159768-75-9 |
Lobradimil (RMP 7)/CAS No.159768-75-9, a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). Lobradimil increases the permeability of the BBB. Lobradimil can be used in the research of brain tumors. |
price> |
R-R-4071 |
R715 CAS No.185052-09-9 |
R715/CAS No.185052-09-9 is a selective bradykinin B1 receptor antagonist. R715 significantly attenuates the hyperalgesic effect developed in Streptozotocin(HY-13753)-diabetic mice. |
price> |
R-R-4072 |
MEN 11270 CAS No.235082-52-7 |
MEN 11270/CAS No.235082-52-7, a cyclic decapeptide, is a B2 kinin receptor antagonist. MEN 11270 bound with high-affinity to the B2 kinin receptor constitutively expressed by WI38 human fibroblasts, inhibiting 3H-bradykinin (BK) with a pKi value of 10.3. |
price> |
R-R-4073 |
Fulimetibant CAS No.2231142-90-6 |
Fulimetibant/CAS No.2231142-90-6 is a bradykinin receptor antagonist. |
price> |
R-R-4074 |
ELN-441958 CAS No.913064-47-8 |
ELN-441958/CAS No.913064-47-8 is a potent, neutral, competitive and selective bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor. ELN-441958 has high oral bioavailability, and has low CNS exposure in the mouse. |
price> |
R-R-4075 |
Bradykinin (2-9) CAS No.16875-11-9 |
Bradykinin (2-9)/CAS No.16875-11-9 is an amino-truncated Bradykinin peptide. Bradykinin (2-9) is a metabolite of Bradykinin, cleaved by Aminopeptidase P. |
price> |
R-R-4076 |
Bradykinin (1-5) CAS No.23815-89-6 |
Bradykinin (1-5)/CAS No.23815-89-6 is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE). |
price> |
R-R-4077 |
[Hyp3]-Bradykinin CAS No.37642-65-2 |
[Hyp3]-Bradykinin/CAS No.37642-65-2, naturally occurring peptide hormone, is a bradykinin receptor agonist. [Hyp3]-Bradykinin interacts with B2-bradykinin receptors and stimulates inositol phosphate production in cultured human fibroblasts. |
price> |
R-R-4078 |
Rimonabant Hydrochloride CAS No.158681-13-1 |
Rimonabant Hydrochloride (SR 141716A Hydrochloride)/CAS No.158681-13-1 is a highly potent and selective central cannabinoid receptor (CB1) antagonist with an Ki of 1.8 nM. Rimonabant Hydrochloride (SR 141716A Hydrochloride) also inhibits Mycobacterial membrane protein Large 3 (MMPL3). |
price> |