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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4063 BIM 23042 TFA BIM 23042 TFA, a certain somatostatin (SS) octapeptide analogue, is a selective neuropeptide neuromedin B receptor (NMB-R, BB1) antagonist. BIM 23042 has 100-fold lower affinity for gastrin-releasing peptide (GRP) receptor (BB2). BIM 23042 inhibits Neuromedin B (HY-P0241), ICI 216140 and DPDM-bombesin ethylamide-induced Ca2+ release. price>
R-R-4064 PD 168368 CAS No.204066-82-0 PD 168368/CAS No.204066-82-0 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with the Ki of 15–45 nM. PD 168368 is neuromedin B receptor (NMBR; IC50=96 nM) / gastrin-releasing peptide receptor (GRPR IC50=3500 nM) antagonist. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC50s of 0.57, 0.24, and 2.7 nM, respectively. price>
R-R-4065 Kuwanon G CAS No.75629-19-5 Kuwanon G/CAS No.75629-19-5 is a flavonoid isolated from Morus alba, acts as a bombesin receptor antagonist, with potential antimicrobial activity. price>
R-R-4066 Kuwanon H CAS No.76472-87-2 Kuwanon H/CAS No.76472-87-2 is a flavonoid isolated from Morus alba, which acts as a potent non-peptide bombesin receptor antagonist. Kuwanon H selectively inhibits binding of gastrin releasing peptide CRP to GRP-preferring recepotr, with a Ki value of 290 nM in cells. price>
R-R-4067 Bradykinin CAS No.58-82-2 Bradykinin/CAS No.58-82-2 is an active peptide that is generated by the kallikrein-kinin system. It is a inflammatory mediator and also recognized as a neuromediator and regulator of several vascular and renal functions. price>
R-R-4068 Icatibant CAS No.130308-48-4 Icatibant (HOE-140)/CAS No.130308-48-4 is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively. price>
R-R-4069 Icatibant acetate CAS No.138614-30-9 Icatibant acetate (HOE-140 acetate)/CAS No.138614-30-9 is a potent and specific peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively. price>
R-R-4070 Lobradimil CAS No.159768-75-9 Lobradimil (RMP 7)/CAS No.159768-75-9, a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). Lobradimil increases the permeability of the BBB. Lobradimil can be used in the research of brain tumors. price>
R-R-4071 R715 CAS No.185052-09-9 R715/CAS No.185052-09-9 is a selective bradykinin B1 receptor antagonist. R715 significantly attenuates the hyperalgesic effect developed in Streptozotocin(HY-13753)-diabetic mice. price>
R-R-4072 MEN 11270 CAS No.235082-52-7 MEN 11270/CAS No.235082-52-7, a cyclic decapeptide, is a B2 kinin receptor antagonist. MEN 11270 bound with high-affinity to the B2 kinin receptor constitutively expressed by WI38 human fibroblasts, inhibiting 3H-bradykinin (BK) with a pKi value of 10.3. price>