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Catalog name Description price
R-R-3893 Tizanidine CAS No.51322-75-9 Tizanidine/CAS No.51322-75-9 is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. price>
R-R-3894 Harmane-d Harmane-d is the deuterium labeled Harmane. Harmane, a β-Carboline alkaloid (BCA), is a potent neurotoxin that causes severe action tremors and psychiatric manifestations. Harmane shows 1000-fold selectivity for I1-Imidazoline receptor (IC50=30 nM) over α2-adrenoceptor (IC50=18 μM). Harmane is also a potent and selective inhibitor of monoamine oxidase (MAO) (IC50s=0.5 and 5 μM for human MAO A/B, respectively). price>
R-R-3895 Tizanidine-d4 CAS No.1188331-19-2 Tizanidine-d4/CAS No.1188331-19-2 is the deuterium labeled Tizanidine. Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. price>
R-R-3896 Metoprolol-d7 hydrochloride CAS No.1219798-61-4 Metoprolol-d7 (hydrochloride)/CAS No.1219798-61-4 is the deuterium labeled Metoprolol. Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties. price>
R-R-3897 Prazosin-d8 CAS No.1006717-55-0 Prazosin-d8/CAS No.1006717-55-0 is the deuterium labeled Prazosin. Prazosin is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder. price>
R-R-3898 Brombuterol-d9 CAS No.1353940-55-2 Brombuterol-d9/CAS No.1353940-55-2 is a deuterium labeled Brombuterol. Brombuterol is a β-adrenergic receptor agonist. price>
R-R-3899 Mibenratide CAS No.1239011-83-6 Mibenratide/CAS No.1239011-83-6, a small cyclic peptide, is an adrenergic β1 receptor antagonist. Mibenratide can be used for heart failure research. price>
R-R-3900 Nadolol-d9 CAS No.94513-92-5 Nadolol-d9/CAS No.94513-92-5 is the deuterium labeled Nadolol. Nadolol is a non-selective and orally active β-adrenergic receptors blocker. price>
R-R-3901 Clorprenaline CAS No.3811-25-4 Clorprenaline/CAS No.3811-25-4 is a potent agonist of β2-adrenergic. Clorprenaline promotes animal muscular mass growth and decreases fat accumulation. Clorprenaline is a potential new lean meat-boosting feed additive. price>
R-R-3902 Salmeterol-d3 CAS No.497063-94-2 Salmeterol-d3/CAS No.497063-94-2 is a deuterium labeled Salmeterol. Salmeterol is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively. price>