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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3861 BMS-466442 CAS No.1598424-76-0 BMS-466442/CAS No.1598424-76-0 is a potent and selective inhibitor of asc-1 (alanine serine cysteine transporter-1), with an IC50 of 11 nM. BMS-466442 inhibits [3H] D-serine uptake into rat brain synaptosomes, with an IC50 of 400 nM. BMS-466442 can be used for schizophrenia research. price>
R-R-3862 Desglymidodrine CAS No.3600-87-1 Desglymidodrine (ST 1059)/CAS No.3600-87-1, the active metabolite of Midodrine (HY-12749), is a selective α1-adrenoceptor agonist. Desglymidodrine is an effective arterial and venous vasoconstrictor and can be used to regulate blood pressure. price>
R-R-3863 Metipranolol hydrochloride CAS No.36592-77-5 Metipranolol hydrochloride/CAS No.36592-77-5 is a non-selective β adrenergic receptor blocking agent. price>
R-R-3864 Dicentrine CAS No.517-66-8 Dicentrine/CAS No.517-66-8 is a natural product isolated from the plant Stephania epigaea Lo with antihypertensive effect. Dicentrine is an α1-adrenoceptor antagonist which has effective against human hyperplastic prostates. price>
R-R-3865 HOKU-81 CAS No.58020-43-2 HOKU-81 (4-Hydroxytulobuterol)/CAS No.58020-43-2 is one of the metabolites of Tulobuterol (HY-B1810). HOKU-81 is a potent and selective β2-adrenoceptor stimulant. HOKU-81 has bronchodilating effect. price>
R-R-3866 (S)-Carvedilol CAS No.95094-00-1 (S)-Carvedilol/CAS No.95094-00-1, the S-enantiomer of Carvedilol, is a non-selective β/α-1 blocker. (S)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX). price>
R-R-3867 FFN270 hydrochloride CAS No.2341841-05-0 FFN270 hydrochloride/CAS No.2341841-05-0, a fluorescent tracer of norepinephrine, is a fluorescent substrate of the norepinephrine and vesicular monoamine transporters. FFN270 hydrochloride exhibits two resolved absorption/excitation maxima depending on solvent pH (FFN270 ex: 320 nm or 365 nm, em: 475 nm) and can function as ratiometric fluorescent pH-sensors. price>
R-R-3892 Levobetaxolol hydrochloride CAS No.116209-55-3 Levobetaxolol hydrochloride/CAS No.116209-55-3 is a beta-adrenergic receptor inhibitor (beta blocker) that can lower the pressure in the eye. price>
R-R-3893 Tizanidine CAS No.51322-75-9 Tizanidine/CAS No.51322-75-9 is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. price>
R-R-3894 Harmane-d Harmane-d is the deuterium labeled Harmane. Harmane, a β-Carboline alkaloid (BCA), is a potent neurotoxin that causes severe action tremors and psychiatric manifestations. Harmane shows 1000-fold selectivity for I1-Imidazoline receptor (IC50=30 nM) over α2-adrenoceptor (IC50=18 μM). Harmane is also a potent and selective inhibitor of monoamine oxidase (MAO) (IC50s=0.5 and 5 μM for human MAO A/B, respectively). price>