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Catalog name Description price
R-R-3813 (+)-Penbutolol CAS No.38363-41-6 (+)-Penbutolol/CAS No.38363-41-6 is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM. (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action. price>
R-R-3814 Todralazine hydrochloride CAS No.3778-76-5 Todralazine hydrochloride (Ecarazine hydrochloride)/CAS No.3778-76-5 is an anti-hypertensive agent, acts as a β2AR blocker, with antioxidant and free radical scavenging activity. price>
R-C-2115 LML-134 CAS：1542135-76-1 LML134(compound 18b)is an orally active and high selective Histamine 3 receptor (H3R)inverse agonist with Kis of 0.3nM and 12nM for hH3R cAMP and hH3R bdg. LML134 penetrates the brain rapidly,leading to high H3R occupancy,and disengages its target with a fast kinetic profile.LML134 has the potential for excessive sleep disorders. price>
R-R-3815 Bufuralol hydrochloride CAS No.60398-91-6 Bufuralol (Ro 3-4787) hydrochloride/CAS No.60398-91-6 is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate. price>
R-R-3816 Tasipimidine sulfate CAS No.1465908-73-9 Tasipimidine sulfate/CAS No.1465908-73-9 is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 against human α2A-adrenoceptor. Tasipimidine sulfate can be used for situational anxiety and fear research. price>
R-R-3817 Propranolol-d7 (ring-d7) CAS No.344298-99-3 Propranolol-d7 (ring-d7)/CAS No.344298-99-3 is the deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively. Propranolol hydrochloride inhibits [3H]-DHA binding to rat brain membrane preparation with an IC50 of 12 nM. Propranolol hydrochloride is used for study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy. price>
R-R-3818 4-Hydroxyatomoxetine CAS No.435293-66-6 4-Hydroxyatomoxetine/CAS No.435293-66-6 is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabolized by the enzyme cytochrome P450 2D6 (CYP2D6). Atomoxetine hydrochloride is a potent and selective noradrenalin re-uptake inhibitor (Ki values are 5 nM, 77 nM and 1451 nM for inhibition of radioligand binding to human NET, SERT and DAT respectively). price>
R-R-3819 Zinterol hydrochloride CAS No.38241-28-0 Zinterol hydrochloride (MJ 9184 hydrochloride)/CAS No.38241-28-0 is a potent and selective β2-adrenoceptor agonist. Zinterol hydrochloride increases ICa in a concentration-dependent manner with an EC50 of 2.2 nM. Zinterol hydrochloride induces ventricular arrhythmias in conscious heart failure rabbits. price>
R-R-3820 A-61603 CAS No.107756-30-9 A-61603/CAS No.107756-30-9 is a selective α1A-adrenergic receptor agonist. A-61603 increases the frequency of spontaneous Ca2+ transients in rat ventricular myocytes in vitro. price>
R-R-3821 Landiolol hydrochloride CAS No.144481-98-1 Landiolol hydrochloride (ONO1101 hydrochloride)/CAS No.144481-98-1 is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity = 255:1, a half-life of 4 min)， acts as an adrenoceptor antagonist. price>