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Catalog name Description price
R-R-3803 Lofexidine hydrochloride CAS No.21498-08-8 Lofexidine (hydrochloride)/CAS No.21498-08-8 is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal. price>
R-C-2104 BAR 502 CAS：1612191-86-2 BAR502 is a dual FXR and GPBAR1 agonist.BAR-502 promotes browning of white adipose tissue and reverses liver steatosis and fibrosis.BAR502 protects against liver damage caused by HFD by promoting the browning of adipose tissue. price>
R-R-3804 Ritodrine hydrochloride CAS No.23239-51-2 Ritodrine (DU21220) hydrochloride/CAS No.23239-51-2 is a β-adrenergic agonist, also an effective smooth muscle and uterine relaxant. Ritodrine hydrochloride prolongs contraction interval, can be used for researching arrest premature labor. price>
R-C-2105 BAR 501 CAS： 1632118-69-4 BAR501 is a potent and selective G protein-coupled bile acid receptor 1(GPBAR1, GPCR19,TGR5)agonist that effectively transactivates GPBAR1 in HEK293 cells overexpressing a CRE along with GPBAR1 with EC50 of 1μM. price>
R-R-3805 Indoramin CAS No.26844-12-2 Indoramin/CAS No.26844-12-2 is an orally active antihypertensive agent. Indoramin is also selective for the α1A-adrenoceptor. price>
R-R-3806 Bucindolol CAS No.71119-11-4 Bucindolol/CAS No.71119-11-4 is a β1-adrenergic receptor blocker, with intrinsic sympathomimetic activity, used in the research of heart failure. price>
R-R-3807 (R)-Terazosin CAS No.109351-34-0 (R)-Terazosin/CAS No.109351-34-0 is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent α1-adrenoceptor antagonist with Ki values of 6.51 nM, 1.01 nM and 1.97 nM for α1a, α1b and α1d-adrenoceptor, respectively. price>
R-R-3808 Phentolamine CAS No.50-60-2 Phentolamine/CAS No.50-60-2 is a potent, selective and orally active α1 adrenergic and α2 adrenergic receptor antagonist. Phentolamine can be used for the research of erectile dysfunction. price>
R-R-3809 (RS)-Butyryltimolol CAS No.2320274-78-8 (RS)-Butyryltimolol/CAS No.2320274-78-8 is the racemate of Butyryltimolol. Butyryltimolol, an effective proagent of Timolol, improves the corneal penetration of Timolol. Butyryltimolol is a β-adrenergic blocker. price>
R-R-3810 Solabegron CAS No.252920-94-8 Solabegron (GW 427353)/CAS No.252920-94-8 is a selective β3-adrenergic receptor agonist, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR, with an EC50 value of 22 nM. Solabegron (GW 427353) is being developed for the treatment of overactive bladder and irritable bowel syndrome. price>