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Catalog name Description price
R-R-3820 A-61603 CAS No.107756-30-9 A-61603/CAS No.107756-30-9 is a selective α1A-adrenergic receptor agonist. A-61603 increases the frequency of spontaneous Ca2+ transients in rat ventricular myocytes in vitro. price>
R-R-3821 Landiolol hydrochloride CAS No.144481-98-1 Landiolol hydrochloride (ONO1101 hydrochloride)/CAS No.144481-98-1 is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity = 255:1, a half-life of 4 min)， acts as an adrenoceptor antagonist. price>
R-R-3822 Meranzin CAS No.23971-42-8 Meranzin/CAS No.23971-42-8 is an absorbed bioactive compound from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS). Meranzin, isolated from leaves of Murraya exotica L., regulates the shared alpha 2-adrenoceptor and involves the AMPA-ERK1/2–BDNF signaling pathway. Meranzin has the potential for the prevention of the comorbidity of atherosclerosis and depression. price>
R-C-2123 LIT-001  CAS： 2245072-21-1 LIT-001 is the first nonpeptide oxytocin receptor(OT-R)agonist(EC50=55 nM;Ki=226nM).LIT-001 improves social interaction in a mouse model of autism. price>
R-C-2125 INCB8761(PF-4136309) CAS：1341224-83-6 PF-4136309(INCB8761)is a potent,selective,and orally bioavailable antagonist of C-C chemokine receptor type 2(CCR2 or CD192(cluster of differentiation 192)with IC50 of 5.2nM,17nM and 13nM for human,mouse and rat CCR2,respectively. price>
R-R-3852 (S)-Terazosin CAS No.109351-33-9 (S)-Terazosin/CAS No.109351-33-9 is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity α-adrenoceptor antagonist with Ki values of 3.91 nM, 0.79 nM and 1.16 nM for α1a, α1b and α1d-adrenoceptor, respectively. (S)-Terazosin also has high-affinity for α2a, α2B and α2c-adrenoceptor with Ki values of 729 nM, 3.5 nM and 46.4 nM, respectively. price>
R-R-3853 Amibegron hydrochloride CAS No.121524-09-2 Amibegron hydrochloride/CAS No.121524-09-2 is a selective β3-adrenoceptor agonist, with an EC50 of 3.5 nM for β-adrenoceptor in rat colon; Amibegron hydrochloride has anxiolytic and antidepressant activity. price>
R-R-3854 Lusaperidone CAS No.214548-46-6 Lusaperidone (R107474)/CAS No.214548-46-6 is an α2 adrenergic receptor antagonist with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively. price>
R-R-3855 ADRA1D receptor antagonist 1 CAS No.1191908-14-1 ADRA1D receptor antagonist 1/CAS No.1191908-14-1 is a potent, selective and orally active α1D adrenoceptor antagonist, with a Ki of 1.6 nM. price>
R-R-3856 Propranolol-d7 CAS No.98897-23-5 Propranolol-d7/CAS No.98897-23-5 is the deuterium labeled Propranolol. Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively. Propranolol inhibits [3H]-DHA binding to rat brain membrane preparation with an IC50 of 12 nM. Propranolol is used for the study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy. price>