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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3794 CGP 20712 A CAS No.105737-62-0 CGP 20712 A (CGP 20712 mesylate)/CAS No.105737-62-0 is a highly selective β1-adrenoceptor antagonist with an IC50 of 0.7 nM. CGP 20712 A exhibits ~10,000-fold selectivity over β2-adrenoceptors. price>
R-R-3795 ONO-2952 CAS No.895169-20-7 ONO-2952/CAS No.895169-20-7 is a potent, selective and orally active translocator protein 18 kDa (TSPO) antagonist with Ki of 0.33-9.30 nM for rat and human TSPO. ONO-2952 is more selective for TSPO than other receptors, transporters, ion channels and enzymes. ONO-2952 exerts its anti-stress effects through inhibition of excessive activation of noradrenergic system in the brain without the amnesic effect. ONO-2952 has the potential for irritable bowel syndrome treatment. price>
R-R-3796 Centanafadine hydrochloride CAS No.923981-14-0 Centanafadine (hydrochloride)/CAS No.923981-14-0 is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively. price>
R-R-3797 Vanilpyruvic acid CAS No.1081-71-6 Vanilpyruvic acid/CAS No.1081-71-6 is a catecholamine metabolite and precursor to vanillactic acid. price>
R-R-3798 Clorprenaline hydrochloride CAS No.6933-90-0 Clorprenaline hydrochloride/CAS No.6933-90-0 is a β2-adrenergic receptor agonist that is implicated in bronchial expansion. Clorprenaline has the potential for asthma research. price>
R-R-3799 Guanadrel CAS No.40580-59-4 Guanadrel/CAS No.40580-59-4 is an orally active postganglionic adrenergic inhibitor of spiroketal. Guanadre can be used in anti-hypertensive studies. price>
R-R-3800 LY377604 CAS No.204592-94-9 LY377604/CAS No.204592-94-9 is a human β3-adrenergic receptor agonist with an EC50 of 2.4 nM and also a β1- and β2-adrenergic receptor antagonist. price>
R-C-2101 BAY-545 CAS：1699717-32-2 BAY-545 is a potent and selective A2B adenosine receptor antagonist, with an IC50 of 59 nM. BAY-545 also exhibits IC50s of 66,400,280 nM for human, mouse,rat A2B adenosine receptor in cells,respectively,and a Ki of 97nM for human A2B adenosine receptor,with more selectivity over A1,A2A,and A3 adenosine receptor. price>
R-R-3801 Apraclonidine hydrochloride CAS No.73218-79-8 Apraclonidine hydrochloride (ALO 2145)/CAS No.73218-79-8, a selective α2 and weak α1 receptor agonist activity, effectively lowers intraocular pressure (IOP) in human eyes. Apraclonidine hydrochloride is a topical ophthalmic solution and has the ability to elevate the eye lid. price>
R-R-3802 Tizanidine hydrochloride CAS No.64461-82-1 Tizanidine hydrochloride/CAS No.64461-82-1 is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. price>