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Catalog name Description price
R-R-3777 Medetomidine CAS No.86347-14-0 Medetomidine/CAS No.86347-14-0 is an orally active α2-adrenoceptor agonist (Ki: 1.08 nM). Medetomidine has sedative and analgesic effects. Medetomidine can cause peripheral vasoconstriction through the activation of α2 adrenoceptors on blood vessels. price>
R-R-3778 Bevantolol hydrochloride CAS No.42864-78-8 Bevantolol hydrochloride/CAS No.42864-78-8 is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist. price>
R-C-2079 E-7046 CAS：1369489-71-3 E7046 is an orally bioavailable and specific EP4 antagonist,with IC50 of 13.5nM and Ki of 23.14nM,exhibiting anti-tumor activities. price>
R-R-3779 Bambuterol hydrochloride CAS No.81732-46-9 Bambuterol hydrochloride/CAS No.81732-46-9 ((±)-Bambuterol hydrochloride; KWD-2183 hydrochloride) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline. price>
R-R-3780 Dabuzalgron CAS No.219311-44-1 Dabuzalgron (Ro 115-1240)/CAS No.219311-44-1 is an orally active and selective α-1A adrenergic receptor agonist for the treatment of urinary incontinence. Dabuzalgron protects against Doxorubicin-induced cardiotoxicity by preserving mitochondrial function. price>
R-C-2081 CPI-444 CAS：1202402-40-1 Ciforadenant(CPI-444,V81444)is a potent and selective Adenosine A2A receptor antagonist.It binds to A2A receptors with a Ki of 3.54 nmol/L and demonstrates a greater than 50-fold selectivity for the A2A receptor over other adenosine receptor subtypes. price>
R-R-3781 Esmolol hydrochloride CAS No.81161-17-3 Esmolol hydrochloride/CAS No.81161-17-3 is a beta adrenergic receptor blocker. price>
R-R-3782 Glaucine CAS No.475-81-0 Glaucine (O,O-Dimethylisoboldine)/CAS No.475-81-0 is an alkaloid isolated from Glaucium flavum with antitussive, bronchodilation and anti-inflammatory properties. Glaucine is a selective and orally active phosphodiesterase 4 (PDE4) inhibitor with Kis of 3.4 µM in human bronchus and polymorphonuclear leukocytes. Glaucine is also a non-selective α-adrenoceptor antagonist, a Ca2+ entry blocker, and a weak dopamine D1 and D2 receptor antagonist. Glaucine has antioxidative and antiviral activities. price>
R-R-3783 Detomidine hydrochloride CAS No.90038-01-0 Detomidine hydrochloride/CAS No.90038-01-0, an imidazole derivative, is a potent α2-adrenergic agonist. Detomidine hydrochloride produces dose-dependent analgesic effects. price>
R-R-3784 Hydrocortisone 17-butyrate CAS No.13609-67-1 Hydrocortisone 17-butyrate/CAS No.13609-67-1 is an adrenocortical hormone active molecule. price>