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Catalog name Description price
R-C-2037 QS11 CAS：944328-88-5 QS11 is an inhibitor of ARFGAP1(ADP-ribosylation factor GTPase-activating protein 1),with an EC50 of 1.5µM.QS11 modulates Wnt/β-catenin signaling through an effect on protein trafficking.QS11 inhibits migration of ARFGAP overexpressing breast cancer cells. price>
R-C-2044 ML-109  CAS：1186649-91-1 ML-109 is a potent and full thyroid stimulating hormone receptor(TSHR)agonist, with an EC50 of 40nM. price>
R-C-2054 JDTIC CAS:361444-66-8 JDTic is a highly selective antagonist for the κ-opioid receptor;without affecting the μ-or δ-opioid receptors. price>
R-R-3774 Terazosin hydrochloride CAS No.63074-08-8 Terazosin hydrochloride/CAS No.63074-08-8 is a quinazoline derivative and a competitive and orally active α1-adrenoceptor antagonist. Terazosin hydrochloride works by relaxing blood vessels and the opening of the bladder. Terazosin hydrochloride has the potential for benign prostatic hyperplasia (BPH) and high blood pressure treatment. price>
R-R-3775 Levobunolol hydrochloride CAS No.27912-14-7 Levobunolol (l-Bunolol) hydrochloride/CAS No.27912-14-7 is a potent and nonselective β-adrenergic receptor antagonist. Levobunolol hydrochloride is an ocular hypotensive agent and lowers mean intraocular pressure (IOP). Levobunolol hydrochloride can be used for glaucoma and superior oblique myokymia (SOM) research. price>
R-R-3776 Isoferulic acid CAS No.537-73-5 Isoferulic acid (3-Hydroxy-4-methoxycinnamic acid)/CAS No.537-73-5 is a cinnamic acid derivative that has antidiabetic activity. Isoferulic acid binds to and activates α1-adrenergic receptors (IC50=1.4 µM) to enhance secretion of β-endorphin (EC50=52.2 nM) and increase glucose use. Isoferulic acid also has anti-influenza virus activities. price>
R-R-3777 Medetomidine CAS No.86347-14-0 Medetomidine/CAS No.86347-14-0 is an orally active α2-adrenoceptor agonist (Ki: 1.08 nM). Medetomidine has sedative and analgesic effects. Medetomidine can cause peripheral vasoconstriction through the activation of α2 adrenoceptors on blood vessels. price>
R-R-3778 Bevantolol hydrochloride CAS No.42864-78-8 Bevantolol hydrochloride/CAS No.42864-78-8 is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist. price>
R-C-2079 E-7046 CAS：1369489-71-3 E7046 is an orally bioavailable and specific EP4 antagonist,with IC50 of 13.5nM and Ki of 23.14nM,exhibiting anti-tumor activities. price>
R-R-3779 Bambuterol hydrochloride CAS No.81732-46-9 Bambuterol hydrochloride/CAS No.81732-46-9 ((±)-Bambuterol hydrochloride; KWD-2183 hydrochloride) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline. price>