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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-C-2021 MK-7246 CAS：1218918-62-7 MK-7246 is a potent and selective CRTH2(chemoattractant receptor-homologous molecule expressed on T-helper type 2 cells)antagonist.MK-7246 is used for the treatment of respiratory diseases. price>
R-C-2025 AMG 837 CAS:865231-46-5 AMG 837 is a potent GPR40 agonist(EC50=13nM)with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. price>
R-C-2026 Nastorazepide CAS:209219-38-5 Nastorazepide(Z-360)is a selective,orally available,1,5-benzodiazepine-derivative gastrin/cholecystokinin 2(CCK-2)receptor antagonist with potential antineoplastic activity. price>
R-C-2034 PIPERIDOLATE CAS：82-98-4 Piperidolate is an antimuscarinic,inhibits intestinal cramp induced by acetylcholine(rats and dogs). price>
R-C-2037 QS11 CAS：944328-88-5 QS11 is an inhibitor of ARFGAP1(ADP-ribosylation factor GTPase-activating protein 1),with an EC50 of 1.5µM.QS11 modulates Wnt/β-catenin signaling through an effect on protein trafficking.QS11 inhibits migration of ARFGAP overexpressing breast cancer cells. price>
R-C-2044 ML-109  CAS：1186649-91-1 ML-109 is a potent and full thyroid stimulating hormone receptor(TSHR)agonist, with an EC50 of 40nM. price>
R-C-2054 JDTIC CAS:361444-66-8 JDTic is a highly selective antagonist for the κ-opioid receptor;without affecting the μ-or δ-opioid receptors. price>
R-R-3774 Terazosin hydrochloride CAS No.63074-08-8 Terazosin hydrochloride/CAS No.63074-08-8 is a quinazoline derivative and a competitive and orally active α1-adrenoceptor antagonist. Terazosin hydrochloride works by relaxing blood vessels and the opening of the bladder. Terazosin hydrochloride has the potential for benign prostatic hyperplasia (BPH) and high blood pressure treatment. price>
R-R-3775 Levobunolol hydrochloride CAS No.27912-14-7 Levobunolol (l-Bunolol) hydrochloride/CAS No.27912-14-7 is a potent and nonselective β-adrenergic receptor antagonist. Levobunolol hydrochloride is an ocular hypotensive agent and lowers mean intraocular pressure (IOP). Levobunolol hydrochloride can be used for glaucoma and superior oblique myokymia (SOM) research. price>
R-R-3776 Isoferulic acid CAS No.537-73-5 Isoferulic acid (3-Hydroxy-4-methoxycinnamic acid)/CAS No.537-73-5 is a cinnamic acid derivative that has antidiabetic activity. Isoferulic acid binds to and activates α1-adrenergic receptors (IC50=1.4 µM) to enhance secretion of β-endorphin (EC50=52.2 nM) and increase glucose use. Isoferulic acid also has anti-influenza virus activities. price>