Products classification
ABOUT US
Email:
sales@ruixibiotech.com
Tel.:
02988811435
Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3617 Medetomidine hydrochloride CAS No.86347-15-1 Medetomidine hydrochloride/CAS No.86347-15-1 is an orally active α2-adrenoceptor agonist (Ki: 1.08 nM). Medetomidine hydrochloride has sedative and analgesic effects. Medetomidine hydrochloride can cause peripheral vasoconstriction through the activation of α2 adrenoceptors on blood vessels. price>
R-R-3618 2-Methoxyidazoxan monohydrochloride CAS No.109544-45-8 2-Methoxyidazoxan monohydrochloride (RX821002 hydrochloride)/CAS No.109544-45-8 is a highly selective alpha 2-adrenoceptor antagonist with little or no imidazoline antagonist effect. RX 821002 has markedly higher affinity for (guinea-pig) alpha 2D-adrenoceptors (pKd 9.7) than for (rabbit) alpha 2A-adrenoceptors (pKd 8.2). price>
R-R-3619 (R)-Carvedilol CAS No.95093-99-5 (R)-Carvedilol ((R)-BM 14190)/CAS No.95093-99-5, the R-enantiomer of Carvedilol, is a non-selective β/α-1 blocker. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX). price>
R-R-3620 Lubabegron CAS No.391920-32-4 Lubabegron/CAS No.391920-32-4 is a potent modulator of β-adrenergic receptor (β -AR). Lubabegron demonstrates antagonistic behavior at the β1 and β 2 receptor subtypes and agonistic behavior at the β 3 receptor subtype in cattle. Lubabegron reduces NH3 gas emissions from an animal or its waste. price>
R-R-3621 Prazosin CAS No.19216-56-9 Prazosin/CAS No.19216-56-9 is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder. price>
R-R-3622 Levonordefrin CAS No.829-74-3 Levonordefrin/CAS No.829-74-3, a common alternative to levoepinephrine as a vasoconstrictor in dental local anesthetic preparations, is usually used in fivefold higher concentrations. Levonordefrin is generally considered equivalent to epinephrine. price>
R-R-3623 Practolol CAS No.6673-35-4 Practolol/CAS No.6673-35-4 is a potent and selective β1-adrenergic receptor antagonist. Practolol can be used for the research of cardiac arrhythmias. price>
R-R-3624 Salmeterol xinafoate CAS No.94749-08-3 Salmeterol (GR 33343X) xinafoate/CAS No.94749-08-3 is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively. price>
R-R-3625 Olodaterol hydrochloride CAS No.869477-96-3 Olodaterol (BI1744) hydrochloride/CAS No.869477-96-3 is a selective, long acting β2-adrenoceptor (β2-AR) agonist (EC50=0.1 nM and pKi= 9.14 for human β2-adrenoceptor, respectively). Olodaterol can be used for chronic obstructive pulmonary disease (COPD) and pulmonary fibrosis. price>
R-R-3626 Bufuralol CAS No.54340-62-4 Bufuralol (Ro 3-4787)/CAS No.54340-62-4 is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate. price>