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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3620 Lubabegron CAS No.391920-32-4 Lubabegron/CAS No.391920-32-4 is a potent modulator of β-adrenergic receptor (β -AR). Lubabegron demonstrates antagonistic behavior at the β1 and β 2 receptor subtypes and agonistic behavior at the β 3 receptor subtype in cattle. Lubabegron reduces NH3 gas emissions from an animal or its waste. price>
R-R-3621 Prazosin CAS No.19216-56-9 Prazosin/CAS No.19216-56-9 is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder. price>
R-R-3622 Levonordefrin CAS No.829-74-3 Levonordefrin/CAS No.829-74-3, a common alternative to levoepinephrine as a vasoconstrictor in dental local anesthetic preparations, is usually used in fivefold higher concentrations. Levonordefrin is generally considered equivalent to epinephrine. price>
R-R-3623 Practolol CAS No.6673-35-4 Practolol/CAS No.6673-35-4 is a potent and selective β1-adrenergic receptor antagonist. Practolol can be used for the research of cardiac arrhythmias. price>
R-R-3624 Salmeterol xinafoate CAS No.94749-08-3 Salmeterol (GR 33343X) xinafoate/CAS No.94749-08-3 is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively. price>
R-R-3625 Olodaterol hydrochloride CAS No.869477-96-3 Olodaterol (BI1744) hydrochloride/CAS No.869477-96-3 is a selective, long acting β2-adrenoceptor (β2-AR) agonist (EC50=0.1 nM and pKi= 9.14 for human β2-adrenoceptor, respectively). Olodaterol can be used for chronic obstructive pulmonary disease (COPD) and pulmonary fibrosis. price>
R-R-3626 Bufuralol CAS No.54340-62-4 Bufuralol (Ro 3-4787)/CAS No.54340-62-4 is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate. price>
R-R-3627 Betaxolol hydrochloride CAS No.63659-19-8 Betaxolol Hydrochloride/CAS No.63659-19-8 is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma. price>
R-C-1929 AM966  CAS：1228690-19-4 AM966 is a high affinity,selective,oral LPA1-antagonist,inhibits LPA-stimulated intracellular calcium release(IC50=17nM). price>
R-C-1930 AM095 CAS: 1228690-36-5 AM095 is a potent LPA1 receptor antagonist because it inhibited GTPγS binding to Chinese hamster ovary(CHO)cell membranes overexpressing recombinant human or mouse LPA1 with IC50 values of 0.98 and 0.73μM,respectively,and exhibited no LPA1 agonism.Lysophosphatidic acid(LPA)is a bioactive phospholipid that signals through a family of at least six G protein-coupled receptors designated LPA1-6. LPA type 1 receptor(LPA1)exhibits widespread tissue distribution and regulates a variety of physiological and pathological cellular functions. price>