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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3615 Penbutolol sulfate CAS No.38363-32-5 Penbutolol sulfate/CAS No.38363-32-5 is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making it a non-selective β blocker. price>
R-R-3616 JP1302 dihydrochloride CAS No.1259314-65-2 JP1302 dihydrochloride/CAS No.1259314-65-2 is a potent, selective, high affinity antagonist of the α2C-adrenoceptor, with a Kb of 16 nM and a Ki of 28 nM for the human α2C-receptor. JP1302 dihydrochloride shows antidepressant and antipsychotic-like effects. JP1302 dihydrochloride can be used for neuropsychiatric disorders and renal dysfunction research. price>
R-R-3617 Medetomidine hydrochloride CAS No.86347-15-1 Medetomidine hydrochloride/CAS No.86347-15-1 is an orally active α2-adrenoceptor agonist (Ki: 1.08 nM). Medetomidine hydrochloride has sedative and analgesic effects. Medetomidine hydrochloride can cause peripheral vasoconstriction through the activation of α2 adrenoceptors on blood vessels. price>
R-R-3618 2-Methoxyidazoxan monohydrochloride CAS No.109544-45-8 2-Methoxyidazoxan monohydrochloride (RX821002 hydrochloride)/CAS No.109544-45-8 is a highly selective alpha 2-adrenoceptor antagonist with little or no imidazoline antagonist effect. RX 821002 has markedly higher affinity for (guinea-pig) alpha 2D-adrenoceptors (pKd 9.7) than for (rabbit) alpha 2A-adrenoceptors (pKd 8.2). price>
R-R-3619 (R)-Carvedilol CAS No.95093-99-5 (R)-Carvedilol ((R)-BM 14190)/CAS No.95093-99-5, the R-enantiomer of Carvedilol, is a non-selective β/α-1 blocker. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX). price>
R-R-3620 Lubabegron CAS No.391920-32-4 Lubabegron/CAS No.391920-32-4 is a potent modulator of β-adrenergic receptor (β -AR). Lubabegron demonstrates antagonistic behavior at the β1 and β 2 receptor subtypes and agonistic behavior at the β 3 receptor subtype in cattle. Lubabegron reduces NH3 gas emissions from an animal or its waste. price>
R-R-3621 Prazosin CAS No.19216-56-9 Prazosin/CAS No.19216-56-9 is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder. price>
R-R-3622 Levonordefrin CAS No.829-74-3 Levonordefrin/CAS No.829-74-3, a common alternative to levoepinephrine as a vasoconstrictor in dental local anesthetic preparations, is usually used in fivefold higher concentrations. Levonordefrin is generally considered equivalent to epinephrine. price>
R-R-3623 Practolol CAS No.6673-35-4 Practolol/CAS No.6673-35-4 is a potent and selective β1-adrenergic receptor antagonist. Practolol can be used for the research of cardiac arrhythmias. price>
R-R-3624 Salmeterol xinafoate CAS No.94749-08-3 Salmeterol (GR 33343X) xinafoate/CAS No.94749-08-3 is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively. price>