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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3903 Guanoxabenz hydrochloride CAS No.23256-40-8 Guanoxabenz (Hydroxyguanabenz) hydrochloride/CAS No.23256-40-8 is an α2 adrenergic receptor agonist, with a Ki of 4000 nM and the fully activated form 40 nM for an α2A adrenoceptor. price>
R-R-3904 Arbutamine CAS No.128470-16-6 Arbutamine/CAS No.128470-16-6 is a short-acting, potent and nonselective β-adrenoceptor agonist. Arbutamine stimulates cardiac β1-, tracheal β2-, and adiopocyte β3- adrenergic receptors. Arbutamine provides cardiac stress increases heart rate, cardiac contractility, and systolic blood pressure. Arbutamine can be used for cardiac stress agent . price>
R-R-3905 Efaroxan hydrochloride CAS No.89197-00-2 Efaroxan hydrochloride/CAS No.89197-00-2 is a potent, selective and orally active α2-adrenoceptor antagonist, with antidiabetic activity. Efaroxan hydrochloride is a selective I1-Imidazoline receptor antagonist. Efaroxan hydrochloride can be used for the research of cardiovascular disease. price>
R-R-3906 NP10679 NP10679 is a selective, pH dependent GluN2B subunit-specific N-methyl-D-aspartate (NMDA) receptor inhibitor with high oral bioavailability and good brain penetration. NP10679 inhibits GluN2B with IC50s of 23 and 142 nM at pH 6.9 and 7.6, respectively. NP10679 is a histamine H1 antagonist and a hERG channel inhibitor with IC50s of 73 and 620 nM, respectively. NP10679 is a reversible inhibitor of human liver CYP enzymes. price>
R-R-3907 Scopine hydrochloride CAS No.85700-55-6 Scopine hydrochloride (6,7-Epoxytropine hydrochloride)/CAS No.85700-55-6 is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock. price>
R-R-3908 Bunazosin CAS No.80755-51-7 Bunazosin/CAS No.80755-51-7 is a potent and selective α1-adrenoceptor antagonist. Bunazosin can be used for antihypertensive and ocular hypotensive research. price>
R-R-3909 Salbutamol-d3 CAS No.1219798-60-3 Salbutamol-d3/CAS No.1219798-60-3 is the deuterium labeled Salbutamol. Salbutamol is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease (COPD). price>
R-R-3910 Midaglizole CAS No.66529-17-7 Midaglizole ((±)-DG5128 free base, DG5128 free base)/CAS No.66529-17-7 is a potent α2-adrenoceptor antagonist. Midaglizole is a hypoglycemic agent. Midaglizole increases blood pressure and reduces blood glucose levels in vivo. price>
R-R-3911 ICI 89406 CAS No.53671-71-9 ICI 89406/CAS No.53671-71-9 is a selective β1 adrenergic receptor antagonist amenable to labelling with positron emitters, for PET. price>
R-R-3912 Phenylephrine-2,4,6-d3 hydrochloride CAS No.1276197-50-2 Phenylephrine-2,4,6-d3 (hydrochloride)/CAS No.1276197-50-2 is the deuterium labeled Phenylephrine hydrochloride. (R)-(-)-Phenylephrine hydrochloride is a selective α1-adrenoceptor agonist with pKis of 5.86, 4.87 and 4.70 for α1D, α1B and α1A receptors respectively. price>