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Catalog name Description price
R-R-3911 ICI 89406 CAS No.53671-71-9 ICI 89406/CAS No.53671-71-9 is a selective β1 adrenergic receptor antagonist amenable to labelling with positron emitters, for PET. price>
R-R-3912 Phenylephrine-2,4,6-d3 hydrochloride CAS No.1276197-50-2 Phenylephrine-2,4,6-d3 (hydrochloride)/CAS No.1276197-50-2 is the deuterium labeled Phenylephrine hydrochloride. (R)-(-)-Phenylephrine hydrochloride is a selective α1-adrenoceptor agonist with pKis of 5.86, 4.87 and 4.70 for α1D, α1B and α1A receptors respectively. price>
R-R-3913 Amosulalol CAS No.85320-68-9 Amosulalol (YM 09538)/CAS No.85320-68-9 is an orally active and dual inhibitor of α1/β1-Adrenergic Receptor. Amosulalol exhibits antihypertensive activity via α1-Adrenergic Receptor inhibition. Amosulalol decreases reflexogenic increases in heart rate and plasma renin activity (PRA) via β1-Adrenergic Receptor inhibition in spontaneously hypertensive rats (SHR). price>
R-R-3914 Yohimbine-13C,d3 CAS No.1261254-59-4 Yohimbine-13C,d3/CAS No.1261254-59-4 is the 13C- and deuterium labeled Yohimbine. Yohimbine is a potent and relatively nonselective alpha 2-adrenergic receptor (AR) antagonist, with IC50 of 0.6 μM. price>
R-R-3915 Upidosin CAS No.152735-23-4 Upidosin (Rec 15/2739)/CAS No.152735-23-4 is an α-1 adrenoceptor (α-1 AR) antagonist. Upidosin shows moderate selectivity for the α-1A AR subtype. Upidosin shows uroselectivity in urethra and prostate with a Kb value of 2-3 nM higher than in ear artery and aorta with a Kb value of 20-100 nM. Upidosin inhibits [3H]prazosin binding to cloned human α-1A adrenergic receptor. Upidosin can be used for the research of urethral obstruction. price>
R-R-3916 4-Hydroxyatomoxetine-d3 CAS No.1217686-14-0 4-Hydroxyatomoxetine-d3/CAS No.1217686-14-0 is a deuterium labeled 4-Hydroxyatomoxetine. 4-Hydroxyatomoxetine is an active metabolite of Atomoxetine (Tomoxetine). 4-Hydroxyatomoxetine is metabolized by the enzyme cytochrome P450 2D6 (CYP2D6). Atomoxetine is a potent and selective noradrenal in re-uptake inhibitor. price>
R-R-3917 Bambuterol-d9 hydrochloride CAS No.1794810-59-5 Bambuterol-d9 (hydrochloride)/CAS No.1794810-59-5 is the deuterium labeled Bambuterol. Bambuterol ((±)-Bambuterol) hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a prodrug of terbutaline. price>
R-R-3918 Abanoquil CAS No.90402-40-7 Abanoquil (U-K52046)/CAS No.90402-40-7, an potent and selective α-1 adrenoceptor antagonist, is an anti-arrhythmic agent. Abanoquil can be used for erectile dysfunction research. price>
R-R-3919 Ivabradine-d6 hydrochloride CAS No.2070009-63-9 Ivabradine-d6 (hydrochloride)/CAS No.2070009-63-9 is the deuterium labeled Ivabradine hydrochloride. Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. price>
R-R-3920 N-(Phenylacetyl-d5)glycine CAS No.1189920-31-7 N-(Phenylacetyl-d5)glycine/CAS No.1189920-31-7 is the deuterium labeled Phenylacetylglycine. Phenylacetylglycine is a gut microbial metabolite that can activate β2AR. Phenylacetylglycine protects against cardiac injury caused by ischemia/reperfusion. price>