Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-2793	[DPro5] Corticotropin Releasing Factor, human, rat TFA	[DPro5] Corticotropin Releasing Factor, human, rat TFA is a selective corticotropin releasing factor/hormone R2 (CRH-R2)agonist. [DPro5] Corticotropin Releasing Factor, human, rat TFA fails to cause the typical anxiogenic effect, but modulates learning and memory processes in rat.	price>
R-R-2794	Stressin I TFA	Stressin I (Cyclo(31-34)[DPhe12,Nle21,38,Glu31,Lys34]Ac-hCRF(4-41)) TFA is a potent CRF1 receptor selective agonist, Ki is 1.7 nM. Stressin I induces an increase in adrenocorticotropic hormone (ACTH) levels in rats.	price>
R-R-2795	Pexacerfont CAS No.459856-18-9	Pexacerfont/CAS No.459856-18-9 is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1±0.6 nM for human CRF1 receptor.	price>
R-R-2796	Antisauvagine-30 TFA	Antisauvagine-30 TFA (aSvg-30 TFA) is a potent, highly selective and competitive CRF2 receptor peptidic antagonist. Antisauvagine-30 TFA exhibits a Kd of 1.4 nM and 150 nM for mCRFR2β and CRFR1, respectively.	price>
R-R-2797	Urocortin III, mouse TFA	Urocortin III, mouse TFA is a corticotropin-releasing factor (CRF)-related peptide. Urocortin III preferentially binds and activates CRF-R2. Urocortin III (Ucn3) is a known component of the behavioral stress response system. Urocortin III and CRF-R2 in the medial amygdala regulate complex social dynamics.	price>
R-R-2798	CP 376395 CAS No.175140-00-8	CP 376395/CAS No.175140-00-8 is a potent, selective, and brain-penetrable Corticotropin releasing factor 1 (CRF1) receptor antagonist.	price>
R-R-2799	DMP 696 CAS No.202578-52-7	DMP 696/CAS No.202578-52-7 is a selective corticotropin-releasing hormone receptor 1 (CRHR1) antagonist, used for the treatment of anxiety and depression.	price>
R-C-1100	Macitentan CAS：441798-33-0	Macitentan is an orally active,non-peptide dual endothelin ETA and ETB receptor antagonist for the potential treatment of idiopathic pulmonary fibrosis(IPF)and pulmonary arterial hypertension(PAH).	price>
R-R-2800	Tildacerfont CAS No.1014983-00-6	Tildacerfont/CAS No.1014983-00-6 is a potent and orally active corticotrophin-releasing factor type 1 (CRF1) receptort antagonis. Tildacerfont effectively reduces adrenocorticotropic hormone (ACTH) and adrenal androgen levels. Tildacerfont has favourable safety profile. Tildacerfont can be used for researching congenital adrenal hyperplasia.	price>
R-R-2801	Antalarmin CAS No.157284-96-3	Antalarmin/CAS No.157284-96-3 is a selective nonpeptide corticotropin-releasing factor receptor 1 (CRHR1) antagonist with a Ki of 2.7 nM. Antalarmin can pass through the blood–brain barrier.	price>

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