Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-2800	Tildacerfont CAS No.1014983-00-6	Tildacerfont/CAS No.1014983-00-6 is a potent and orally active corticotrophin-releasing factor type 1 (CRF1) receptort antagonis. Tildacerfont effectively reduces adrenocorticotropic hormone (ACTH) and adrenal androgen levels. Tildacerfont has favourable safety profile. Tildacerfont can be used for researching congenital adrenal hyperplasia.	price>
R-R-2801	Antalarmin CAS No.157284-96-3	Antalarmin/CAS No.157284-96-3 is a selective nonpeptide corticotropin-releasing factor receptor 1 (CRHR1) antagonist with a Ki of 2.7 nM. Antalarmin can pass through the blood–brain barrier.	price>
R-R-2802	a-Helical CRF(9-41) TFA	α-Helical CRF(9-41) TFA is a competitive CRF2 receptor antagonist with KB of ~100 nM. α-Helical CRF(9-41) TFA is also a partial agonist of CRF1 receptor with an EC50 of 140 nM.	price>
R-R-2803	Urocortin, rat CAS No.171543-83-2	Urocortin, rat (Urocortin (Rattus norvegicus))/CAS No.171543-83-2 is a neuropeptide and a potent endogenous CRFR agonist with Kis of 13 nM, 1.5 nM, and 0.97 nM for human CRF1, rat CRF2α and mouse CRF2β, respectively.	price>
R-R-2804	NBI-27914 hydrochloride CAS No.1215766-76-9	NBI-27914 (hydrochloride)/CAS No.1215766-76-9 is a selective Corticotropin-Releasing Factor 1 (CRF1) receptor antagonist with a Ki value of 1.7 nM.	price>
R-R-2805	Urotensin I TFA	Urotensin I (Catostomus urotensin I) TFA, a CRF-like neuropeptide, acts as an agonist of CRF receptor with pEC50s of 11.46, 9.36 and 9.85 for human CRF1, human CRF2 and rat CRF2α receptors in CHO cells, and Kis of 0.4, 1.8, and 5.7 nM for hCRF1, rCRF2α and mCRF2β receptors, respectively.	price>
R-R-2806	Liraglutide CAS No.204656-20-2	Liraglutide/CAS No.204656-20-2 is a glucagon-like peptide-1 (GLP-1) receptor agonist used clinically to treat type 2 diabetes mellitus.	price>
R-R-2807	NN1177 TFA	NN1177 (NNC9204-1177) TFA is a long-acting GLP-1/glucagon receptor co-agonist. NN1177 TFA can induce a dose-dependent body weight loss in diet-induced obese (DIO) mice.	price>
R-C-1108	ANA-12 CAS： 219766-25-3	ANA-12 is a potent and selective TrkB antagonist with IC50s of 45.6 nM and 41.1 μM for the high and low affinity sites,respectively.	price>
R-R-2808	Emicerfont CAS No.786701-13-1	Emicerfont/CAS No.786701-13-1 is a corticotropin-releasing factor type 1 (CRF1) receptor antagonist with an IC50 of 66 nM.	price>

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