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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4119 RVD-Hpα TFA CAS No.1431329-51-9 RVD-Hpα TFA/CAS No.1431329-51-9 is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM). price>
R-R-4120 BML-190 CAS No.2854-32-2 BML-190(IMMA)/CAS No.2854-32-2 is a potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively). price>
R-R-4121 Auriculasin CAS No.60297-37-2 Auriculasin/CAS No.60297-37-2 is a nature product isolated from Limonium leptophyllum. Auriculasin has activity toward cannabinoid receptor type 1 (CB1) with an IC50 value of 8.92 µM. price>
R-R-4122 Arvanil CAS No.128007-31-8 Arvanil/CAS No.128007-31-8 is a ligand for vanilloid receptor 1 (VR1) and cannabinoid 1 (CB1). Arvanil can inhibit spasticity, as a potent neuroprotectant. price>
R-R-4123 Taranabant ((1R,2R)stereoisomer) CAS No.701977-08-4 Taranabant (1R,2R)stereoisomer/CAS No.701977-08-4 is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. price>
R-R-4124 Drinabant CAS No.358970-97-5 Drinabant (AVE1625)/CAS No.358970-97-5 is an orally active CB1 receptor antagonist. Drinabant (AVE1625) inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R. price>
R-R-4125 CB65 CAS No.913534-05-1 CB65/CAS No.913534-05-1 is a potent and high affinity CB2 selective agonist with a Ki value of 3.3 nM. CB65 exhibits a Ki of >1000 nM for CB1 receptor. price>
R-R-4126 CB2R/FAAH modulator-3 CAS No.2876918-67-9 CB2R/FAAH modulator-3 (compound 27)/CAS No.2876918-67-9 is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-3 are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection. price>
R-R-4127 PGN36 CAS No.1564253-75-3 PGN36 (Compound 18)/CAS No.1564253-75-3 is a selective cannabinoid CB2 receptor (CB2R) antagonist with a Ki of 0.09 µM. price>
R-R-4128 AM6545 CAS No.1245626-05-4 AM6545/CAS No.1245626-05-4 is a peripherally active, cannabinoid receptor antagonist with limited brain penetration. AM6545 binds to CB1 and CB2 receptors with Kis of 1.7 nM and 523 nM, respectively. AM6545 is a neutral antagonist. AM6545 can be used for the research of obesity and its complications. price>