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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4117 JTE-907 CAS No.282089-49-0 JTE-907/CAS No.282089-49-0 is a highly selective, orally active CB2 receptor inverse agonist and exerts anti-inflammatory effects in vivo. price>
R-R-4118 GP1a CAS No.511532-96-0 GP1a/CAS No.511532-96-0 is a potent agonist of cannabinoid receptor 2 (CB2). Gp1a is beneficial to skin wound healing. GP1a inhibits inflammation and fibrogenesis while promoting re-epithelialization. price>
R-C-2419 Droxidopa CAS:23651-95-8 Droxidopa is a synthetic amino acid precursor which acts as a prodrug to the neurotransmitters norepinephrine(noradrenaline)and epinephrine(adrenaline)and it is used to increase the concentrations of these neurotransmitters in the body and brain.Unlike norepinephrine and epinephrine themselves,droxidopa is capable of crossing the protective blood–brain barrier(BBB). price>
R-R-4119 RVD-Hpα TFA CAS No.1431329-51-9 RVD-Hpα TFA/CAS No.1431329-51-9 is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM). price>
R-R-4120 BML-190 CAS No.2854-32-2 BML-190(IMMA)/CAS No.2854-32-2 is a potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively). price>
R-R-4121 Auriculasin CAS No.60297-37-2 Auriculasin/CAS No.60297-37-2 is a nature product isolated from Limonium leptophyllum. Auriculasin has activity toward cannabinoid receptor type 1 (CB1) with an IC50 value of 8.92 µM. price>
R-R-4122 Arvanil CAS No.128007-31-8 Arvanil/CAS No.128007-31-8 is a ligand for vanilloid receptor 1 (VR1) and cannabinoid 1 (CB1). Arvanil can inhibit spasticity, as a potent neuroprotectant. price>
R-R-4123 Taranabant ((1R,2R)stereoisomer) CAS No.701977-08-4 Taranabant (1R,2R)stereoisomer/CAS No.701977-08-4 is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. price>
R-R-4124 Drinabant CAS No.358970-97-5 Drinabant (AVE1625)/CAS No.358970-97-5 is an orally active CB1 receptor antagonist. Drinabant (AVE1625) inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R. price>
R-R-4125 CB65 CAS No.913534-05-1 CB65/CAS No.913534-05-1 is a potent and high affinity CB2 selective agonist with a Ki value of 3.3 nM. CB65 exhibits a Ki of >1000 nM for CB1 receptor. price>