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Catalog name Description price
R-R-3996 Olodanrigan CAS No.1316755-16-4 Olodanrigan (EMA401)/CAS No.1316755-16-4 is a highly selective, orally active, peripherally restricted angiotensin II type 2 receptor (AT2R) antagonist. It is under development as a neuropathic pain therapeutic agent. Olodanrigan (EMA401) analgesic action appears to involve inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hyperexcitability and sprouting of DRG neurons. price>
R-R-3997 PD 123319 ditrifluoroacetate CAS No.136676-91-0 PD 123319 (ditrifluoroacetate)/CAS No.136676-91-0 is a potent, selective AT2 angiotensin II receptor antagonist with IC50 of 34 nM. price>
R-R-3998 Azilsartan medoxomil CAS No.863031-21-4 Azilsartan medoxomil (TAK 491)/CAS No.863031-21-4 is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. price>
R-R-3999 Angiotensin II 5-valine CAS No.58-49-1 Angiotensin II 5-valine/CAS No.58-49-1 is an agonist of angiotensin receptor. price>
R-R-4000 Olmesartan medoxomil CAS No.144689-63-4 Olmesartan medoxomil/CAS No.144689-63-4 is a potent and selective angiotensin AT1 receptor inhibitor with IC50 of 66.2 μM. price>
R-R-4001 Benzyl benzoate CAS No.120-51-4 Benzyl benzoate (Phenylmethyl benzoate)/CAS No.120-51-4 is an orally active anti-scabies agent, acaricide (EC50= 0.06 g/m2) and fungicide. Benzyl benzoate is an angiotensin II (Ang II) inhibitor with antihypertensive effects. Benzyl benzoate can be used in perfumes, pharmaceuticals and the food industry. price>
R-R-4017 TRV055 hydrochloride TRV055 hydrochloride, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 hydrochloride is efficacious in stimulating cellular Gq-mediated signaling. price>
R-R-4018 TRV056 CAS No.812644-79-4 TRV056/CAS No.812644-79-4 is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV056 is efficacious in stimulating cellular Gq-mediated signaling. TRV056 can be used to develop the Gq-biased AT1R agonists. price>
R-R-4019 TRV055 CAS No.25849-90-5 TRV055/CAS No.25849-90-5, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 is efficacious in stimulating cellular Gq-mediated signaling. price>
R-R-4020 Norleual TFA Norleual TFA, an angiotensin (Ang) IV analog, is a hepatocyte growth factor (HGF)/c-Met inhibitor with an IC50 of 3 pM. Norleual TFA is an AT4 receptor antagonist and exhibits potent antiangiogenic activities. price>