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Catalog name Description price
R-R-4001 Benzyl benzoate CAS No.120-51-4 Benzyl benzoate (Phenylmethyl benzoate)/CAS No.120-51-4 is an orally active anti-scabies agent, acaricide (EC50= 0.06 g/m2) and fungicide. Benzyl benzoate is an angiotensin II (Ang II) inhibitor with antihypertensive effects. Benzyl benzoate can be used in perfumes, pharmaceuticals and the food industry. price>
R-R-4017 TRV055 hydrochloride TRV055 hydrochloride, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 hydrochloride is efficacious in stimulating cellular Gq-mediated signaling. price>
R-R-4018 TRV056 CAS No.812644-79-4 TRV056/CAS No.812644-79-4 is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV056 is efficacious in stimulating cellular Gq-mediated signaling. TRV056 can be used to develop the Gq-biased AT1R agonists. price>
R-R-4019 TRV055 CAS No.25849-90-5 TRV055/CAS No.25849-90-5, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 is efficacious in stimulating cellular Gq-mediated signaling. price>
R-R-4020 Norleual TFA Norleual TFA, an angiotensin (Ang) IV analog, is a hepatocyte growth factor (HGF)/c-Met inhibitor with an IC50 of 3 pM. Norleual TFA is an AT4 receptor antagonist and exhibits potent antiangiogenic activities. price>
R-R-4021 GSK1820795A CAS No.2650253-86-2 GSK1820795A/CAS No.2650253-86-2, as a telmisartan analog, is a selective hGPR132a antagonist. GSK1820795A blocks activation of yeast cells expressing hGPR132a by N-acylamides. GSK1820795A is also a angiotensin II antagonists and partial PPARγ agonists (compound 38). price>
R-R-4022 Azilsartan-d5 CAS No.1346599-45-8 Azilsartan-d5/CAS No.1346599-45-8 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. price>
R-R-4023 Irbesartan-d4 CAS No.1216883-23-6 Irbesartan-d4/CAS No.1216883-23-6 is the deuterium labeled Irbesartan, which is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist. price>
R-R-4024 Telmisartan-d3 CAS No.1189889-44-8 Telmisartan-d3/CAS No.1189889-44-8 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM. price>
R-R-4025 Eprosartan mesylate CAS No.144143-96-4 Eprosartan mesylate (SKF-108566J)/CAS No.144143-96-4 is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan mesylate binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively. price>