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Catalog name Description price
R-R-4000 Olmesartan medoxomil CAS No.144689-63-4 Olmesartan medoxomil/CAS No.144689-63-4 is a potent and selective angiotensin AT1 receptor inhibitor with IC50 of 66.2 μM. price>
R-R-4001 Benzyl benzoate CAS No.120-51-4 Benzyl benzoate (Phenylmethyl benzoate)/CAS No.120-51-4 is an orally active anti-scabies agent, acaricide (EC50= 0.06 g/m2) and fungicide. Benzyl benzoate is an angiotensin II (Ang II) inhibitor with antihypertensive effects. Benzyl benzoate can be used in perfumes, pharmaceuticals and the food industry. price>
R-R-4017 TRV055 hydrochloride TRV055 hydrochloride, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 hydrochloride is efficacious in stimulating cellular Gq-mediated signaling. price>
R-R-4018 TRV056 CAS No.812644-79-4 TRV056/CAS No.812644-79-4 is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV056 is efficacious in stimulating cellular Gq-mediated signaling. TRV056 can be used to develop the Gq-biased AT1R agonists. price>
R-R-4019 TRV055 CAS No.25849-90-5 TRV055/CAS No.25849-90-5, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 is efficacious in stimulating cellular Gq-mediated signaling. price>
R-R-4020 Norleual TFA Norleual TFA, an angiotensin (Ang) IV analog, is a hepatocyte growth factor (HGF)/c-Met inhibitor with an IC50 of 3 pM. Norleual TFA is an AT4 receptor antagonist and exhibits potent antiangiogenic activities. price>
R-R-4021 GSK1820795A CAS No.2650253-86-2 GSK1820795A/CAS No.2650253-86-2, as a telmisartan analog, is a selective hGPR132a antagonist. GSK1820795A blocks activation of yeast cells expressing hGPR132a by N-acylamides. GSK1820795A is also a angiotensin II antagonists and partial PPARγ agonists (compound 38). price>
R-R-4022 Azilsartan-d5 CAS No.1346599-45-8 Azilsartan-d5/CAS No.1346599-45-8 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. price>
R-R-4023 Irbesartan-d4 CAS No.1216883-23-6 Irbesartan-d4/CAS No.1216883-23-6 is the deuterium labeled Irbesartan, which is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist. price>
R-R-4024 Telmisartan-d3 CAS No.1189889-44-8 Telmisartan-d3/CAS No.1189889-44-8 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM. price>