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Catalog name Description price
R-R-3976 Isoxsuprine-d6 hydrochloride CAS No.2706004-35-3 Isoxsuprine-d6 (hydrochloride)/CAS No.2706004-35-3 is the deuterium labeled Isoxsuprine hydrochloride. Isoxsuprine hydrochloride is a beta-adrenergic receptor agonist with Kis of 13.65 μΜ and 3.48 μΜ for myometrial and placcntal beta-adrenergic receptor, respectively. Isoxsuprine hydrochloride is also a NMDA receptor antagonist. price>
R-R-3977 Azepexole dihydrochloride CAS No.36067-72-8 Azepexole (B-HT 933) dihydrochloride/CAS No.36067-72-8 is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM). price>
R-R-3978 Betaxolol-d7 hydrochloride CAS No.1219802-92-2 Betaxolol-d7 (hydrochloride)/CAS No.1219802-92-2 is the deuterium labeled Betaxolol hydrochloride. Betaxolol Hydrochloride is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma. price>
R-R-3979 Cimbuterol CAS No.54239-39-3 Cimbuterol/CAS No.54239-39-3 is a β-adrenergic receptor agonist. price>
R-R-3980 Tizanidine-d4 hydrochloride CAS No.1188263-51-5 Tizanidine-d4 (hydrochloride)/CAS No.1188263-51-5 is deuterium labeled Tizanidine (hydrochloride). price>
R-R-3981 Guanfacine-13C,15N3 CAS No.1189924-28-4 Guanfacine-13C,15N3/CAS No.1189924-28-4 is the 13C and 15N labeled Guanfacine. Guanfacine is an orally active noradrenergic α2A agonist and has high selective for the α2A receptor subtype. Guanfacine has effects in producing hypotension and sedation. price>
R-R-3982 Talibegron hydrochloride CAS No.178600-17-4 Talibegron hydrochloride (ZD2079 hydrochloride)/CAS No.178600-17-4 is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect. price>
R-R-3983 Perphenazine-d8 dihydrochloride CAS No.2070015-23-3 Perphenazine-d8 (dihydrochloride)/CAS No.2070015-23-3 is the deuterium labeled Perphenazine, which is a typical antipsychotic agent(5-HT, Dopamine receptor ligand). price>
R-R-3984 Phentolamine-d4 hydrochloride CAS No.1346599-65-2 Phentolamine-d4 (hydrochloride)/CAS No.1346599-65-2 is the deuterium labeled Phentolamine hydrochloride. Phentolamine hydrochloride is a reversible, non-selective, and orally active blocker of α1 and α2 adrenergic receptor that expands blood vessels to reduce peripheral vascular resistance. Phentolamine hydrochloride can be used for the research of pheochromocytoma-related hypertension, heart failure and erectile dysfunction. price>
R-R-3985 Silodosin-d4 CAS No.1426173-86-5 Silodosin-d4/CAS No.1426173-86-5 is the deuterium labeled Silodosin. Silodosin (KAD 3213) is a potent, selective and orally active α1A-adrenergic receptor (α1A-AR) blocker. Silodosin exhibits high affinity for α1A-AR (Ki=0.036 nM), over 162-fold and 50-fold than for α1B-AR and α1D-AR with Ki values of 21 nM and 2.0 nM, respectively. Silodosin is an effective and well-tolerated agent, it can be used for the investigation of LUTS/BPH. price>